SCHEMBL3400915

SCHEMBL3400915

COc1cc(CC(=O)c2ccccc2)sc1C(=O)N1CCC[C@H]1CN1CCCC1

nearest known ligand 0.50

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 12/20 0.50
MET P08581 3/20 0.44
KCNH2 Q12809 2/20 0.43
ITGB1 P05556 1/20 0.41
ITGA4 P13612 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3402115 0.81 HRH3 (0.48) HRH3METKCNH2
SCHEMBL10293592 0.75 HRH3 (0.62) HRH3METKCNH2
SCHEMBL10293596 0.75 HRH3 (0.62) HRH3METKCNH2
SCHEMBL5217166 0.73 HRH3 (0.72) HRH3KCNH2
SCHEMBL17570419 0.72 HRH3 (0.59) HRH3METKCNH2
SCHEMBL12615622 0.72 HRH3 (0.66) HRH3
SCHEMBL12615280 0.72 HRH3 (0.66) HRH3
SCHEMBL2743633 0.71 HRH3 (0.56) HRH3METKCNH2
SCHEMBL2743632 0.71 HRH3 (0.56) HRH3METKCNH2
SCHEMBL2743650 0.71 HRH3 (0.57) HRH3METKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2247588-A2 FUSED HETEROCYCLIC DERIVATIVE AND USE THEREOF Takeda Pharmaceutical Company Limited (JP) 2010-11-10 EP disclosed
WO-2009107850-A2 FUSED HETEROCYCLIC DERIVATIVE AND USE THEREOF TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-09-03 WO disclosed