SCHEMBL3402115

SCHEMBL3402115

COc1cc(Cc2ccccn2)sc1C(=O)N1CCC[C@H]1CN1CCCC1

nearest known ligand 0.48

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 6/20 0.48
POLB P06746 1/20 0.45
HCRTR1 O43613 2/20 0.43
HCRTR2 O43614 2/20 0.43
MET P08581 5/20 0.42
ALDH1A1 P00352 2/20 0.41
KDM4E B2RXH2 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
KCNH2 Q12809 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3400915 0.81 HRH3 (0.50) HRH3METKCNH2
SCHEMBL3274929 0.74 MET (0.53) HRH3POLBMETALDH1A1
SCHEMBL3274932 0.74 MET (0.53) HRH3POLBMETALDH1A1
SCHEMBL3282430 0.74 MET (0.53) HRH3POLBMETALDH1A1
SCHEMBL3275537 0.73 MET (0.48) HRH3METKCNH2
SCHEMBL3275541 0.73 MET (0.48) HRH3METKCNH2
Hydrochloric Acid SCHEMBL3275163 0.73 MET (0.52) HRH3POLBMETALDH1A1
Hydrochloric Acid SCHEMBL3275160 0.73 MET (0.52) HRH3POLBMETALDH1A1
SCHEMBL10314339 0.73 HRH3 (0.46) HRH3POLBHCRTR1HCRTR2ALDH1A1
SCHEMBL3275616 0.71 MET (0.48) HRH3POLBHCRTR1HCRTR2MET

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2247588-A2 FUSED HETEROCYCLIC DERIVATIVE AND USE THEREOF Takeda Pharmaceutical Company Limited (JP) 2010-11-10 EP disclosed
WO-2009107850-A2 FUSED HETEROCYCLIC DERIVATIVE AND USE THEREOF TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-09-03 WO disclosed