SCHEMBL3400970

SCHEMBL3400970

CCn1c(C(=O)N2CCN(C(C)C)CC2)cnc1-c1cccc2ccccc12

nearest known ligand 0.42

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 2/20 0.42
HTR2C P28335 13/20 0.41
HTR2A P28223 1/20 0.41
HRH3 Q9Y5N1 4/20 0.40
LMNA P02545 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3402645 0.86 PARP1 (0.47) PARP1HTR2CHTR2AHRH3
SCHEMBL3403662 0.83 ACACB (0.44) HTR2CHTR2ALMNA
SCHEMBL3402312 0.83 HTR2C (0.43) HTR2CHTR2AHRH3LMNA
SCHEMBL3402101 0.82 HTR2C (0.53) PARP1HTR2CHRH3LMNA
SCHEMBL3405656 0.81 HTR2C (0.45) PARP1HTR2CHRH3LMNA
SCHEMBL3402974 0.79 KDM4E (0.48) HTR2CLMNA
SCHEMBL3399942 0.78 HTR2C (0.42) HTR2CHRH3LMNA
SCHEMBL3402302 0.76 CDC25B (0.46) LMNA
SCHEMBL13310444 0.76 HTR2C (0.37) PARP1HTR2CHRH3LMNA
SCHEMBL3402464 0.74 HTR2C (0.52) PARP1HTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7728009-B1 Thiazole amides, imidazole amides and related analogues NEUROGEN CORPORATION (US) 2010-06-01 US disclosed
US-7728009-B1 Thiazole amides, imidazole amides and related analogues NEUROGEN CORPORATION (US) 2010-06-01 US disclosed
US-7728009-B1 Thiazole amides, imidazole amides and related analogues NEUROGEN CORPORATION (US) 2010-06-01 US disclosed
WO-2006089076-A9 THIAZOLE AMIDES, IMIDAZOLE AMIDES AND RELATED ANALOGUES NEUROGEN CORP (US) 2007-04-26 WO disclosed