SCHEMBL3401136

SCHEMBL3401136

CC(=O)O[C@@H]1[C@@H](OC(C)=O)[C@@H](Oc2cnc(-c3cccnc3)c(F)c2)SC[C@H]1OC(C)=O

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C19 P33261 3/20 0.35
ADORA2B P29275 2/20 0.35
CYP3A4 P08684 2/20 0.34
CYP11B2 P19099 4/20 0.33
HCRTR1 O43613 4/20 0.33
HCRTR2 O43614 4/20 0.33
CYP11B1 P15538 2/20 0.33
CDC7 O00311 1/20 0.32
DBF4 Q9UBU7 1/20 0.32
ALDH1A1 P00352 1/20 0.32
LMNA P02545 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP19A1 P11511 1/20 0.32
ABCB1 P08183 2/20 0.32
CTSA P10619 1/20 0.32
AKR1C3 P42330 1/20 0.31
AKR1C2 P52895 1/20 0.31
ABL1 P00519 1/20 0.31
CYP2A6 P11509 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL315036 1.00 CYP2C19 (0.35) CYP2C19ADORA2BCYP3A4CYP11B2HCRTR1
SCHEMBL2139978 0.91 DHODH (0.35) HCRTR1HCRTR2CTSA
SCHEMBL2139974 0.91 DHODH (0.35) HCRTR1HCRTR2CTSA
SCHEMBL3399355 0.90 ADORA2A (0.32) CYP2C19ADORA2BCYP3A4
SCHEMBL314779 0.90 ADORA2A (0.32) CYP2C19ADORA2BCYP3A4
SCHEMBL3395742 0.90
SCHEMBL314966 0.90
SCHEMBL315234 0.89 FFAR4 (0.33)
SCHEMBL315235 0.89 FFAR4 (0.33)
SCHEMBL314511 0.87 WNT3A (0.34)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2066683-B1 DERIVATIVES OF 5-THIOXYLOPYRANOSE AND USE OF SAME FOR TREATMENT FOURNIER LAB SA (FR) 2010-11-03 EP disclosed