SCHEMBL3401299

SCHEMBL3401299

CCN(CC)C1CCN(C(=O)c2sc(-c3ccc(F)cc3F)nc2C)C1

nearest known ligand 0.48

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ACKR3 P25106 1/20 0.47
HTR2C P28335 7/20 0.44
POLR1A O95602 1/20 0.40
CBX7 O95931 1/20 0.40
CDYL2 Q8N8U2 1/20 0.40
CDYL Q9Y232 1/20 0.40
CDY1; CDY1B Q9Y6F8 1/20 0.40
CES2 O00748 1/20 0.38
PARP1 P09874 1/20 0.38
KDM1A O60341 1/20 0.38
GAA P10253 1/20 0.38
S1PR1 P21453 1/20 0.38
S1PR3 Q99500 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3401129 0.95 ACKR3 (0.50) ACKR3HTR2CCBX7CDYL2CDYL
SCHEMBL3405850 0.94 HTR2C (0.44) ACKR3HTR2CPOLR1ACBX7CDYL2
SCHEMBL3405875 0.92 HTR2C (0.44) ACKR3HTR2CPOLR1ACBX7CDYL2
SCHEMBL3400020 0.88 HTR2C (0.41) ACKR3HTR2CPOLR1A
SCHEMBL3405458 0.88 HTR2C (0.47) ACKR3HTR2CCBX7CDYL2CDYL
SCHEMBL3400092 0.86 HTR2C (0.47) ACKR3HTR2CCBX7CDYL2CDYL
SCHEMBL13310351 0.85 HTR2C (0.46) ACKR3HTR2CCBX7CDYL2CDYL
SCHEMBL3401811 0.84 HTR2C (0.45) HTR2CPOLR1ACES2KDM1A
SCHEMBL3398514 0.84 KDM4E (0.46) HTR2CPOLR1A
SCHEMBL3399783 0.84 HTR2C (0.45) HTR2CPOLR1ACES2KDM1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7728009-B1 Thiazole amides, imidazole amides and related analogues NEUROGEN CORPORATION (US) 2010-06-01 US disclosed
US-7728009-B1 Thiazole amides, imidazole amides and related analogues NEUROGEN CORPORATION (US) 2010-06-01 US disclosed
US-7728009-B1 Thiazole amides, imidazole amides and related analogues NEUROGEN CORPORATION (US) 2010-06-01 US disclosed
WO-2006089076-A9 THIAZOLE AMIDES, IMIDAZOLE AMIDES AND RELATED ANALOGUES NEUROGEN CORP (US) 2007-04-26 WO disclosed