SCHEMBL3401394

SCHEMBL3401394

CCC(Br)n1c2ccccc2c2ccccc21

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPR3 P46089 1/20 0.43
CYP1A2 P05177 1/20 0.41
CYP2C19 P33261 1/20 0.41
POLB P06746 2/20 0.41
BACE1 P56817 2/20 0.39
ALDH1A1 P00352 2/20 0.38
TSHR P16473 2/20 0.38
NPY1R P25929 1/20 0.38
NPY2R P49146 1/20 0.38
MAPT P10636 2/20 0.37
MAPK1 P28482 2/20 0.37
TDP1 Q9NUW8 2/20 0.37
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
KDM4E B2RXH2 2/20 0.37
HPGD P15428 1/20 0.37
HTT P42858 1/20 0.37
HBB P68871 1/20 0.37
HSD17B10 Q99714 1/20 0.37
BCHE P06276 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12027587 0.80 CNR2 (0.42) GPR3CYP1A2CYP2C19ALDH1A1TDP1
SCHEMBL573153 0.78 CYP1A2 (0.50) GPR3CYP1A2CYP2C19POLBBACE1
SCHEMBL12091659 0.78 GPR3 (0.46) GPR3CYP1A2CYP2C19POLBBACE1
SCHEMBL5668880 0.78 CNR1 (0.41) PGRRORARORCRORB
SCHEMBL27749998 0.78 CNR1 (0.41) PGRRORARORCRORB
SCHEMBL28231424 0.78 CNR1 (0.41) PGRRORARORCRORB
SCHEMBL28129667 0.78 CNR1 (0.41) PGRRORARORCRORB
SCHEMBL18404644 0.77 GPR3 (0.44) GPR3CYP1A2CYP2C19POLBBACE1
SCHEMBL14164189 0.77 GPR3 (0.44) GPR3CYP1A2CYP2C19POLBBACE1
SCHEMBL127116 0.77 GPR3 (0.44) GPR3CYP1A2CYP2C19POLBBACE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2231140-A1 SIGMA LIGANDS AND IKK / NF - KB INHIBITORS FOR MEDICAL TREATMENT University of Dundee (GB) 2010-09-29 EP disclosed
WO-2009074809-A1 SIGMA LIGANDS AND IKK / NF - KB INHIBITORS FOR MEDICAL TREATMENT UNIVERSITY OF DUNDEE (GB) 2009-06-18 WO disclosed