SCHEMBL3401452

SCHEMBL3401452

C[CH]CCCN(CC)CC(N)=O

nearest known ligand 0.35

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 1/20 0.35
ALDH1A1 P00352 1/20 0.33
MEN1 O00255 1/20 0.32
FAAH O00519 1/20 0.32
TP53 P04637 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2C19 P33261 1/20 0.32
SOAT1 P35610 1/20 0.32
KMT2A Q03164 1/20 0.32
PAOX Q6QHF9 1/20 0.31
CNR1 P21554 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8417254 0.80 CA12 (0.45) NPSR1ALDH1A1MEN1FAAHTP53
SCHEMBL8383111 0.79 KDM5A (0.41) NPSR1MEN1FAAHTP53CYP1A2
SCHEMBL644835 0.77 SIGMAR1 (0.34) NPSR1ALDH1A1MEN1KMT2APAOX
SCHEMBL8416737 0.76 CA12 (0.39) NPSR1ALDH1A1CYP2C19
SCHEMBL177796 0.75
SCHEMBL18902827 0.75 CHRM2 (0.39) NPSR1ALDH1A1TP53CYP1A2CYP3A4
SCHEMBL3267270 0.74 CHRM2 (0.38) NPSR1ALDH1A1TP53CYP1A2CYP3A4
SCHEMBL8415770 0.73 CA1 (0.33) NPSR1ALDH1A1
Hydrochloric Acid SCHEMBL3453649 0.73 CHRM2 (0.38) NPSR1ALDH1A1TP53CYP1A2CYP3A4
SCHEMBL13895313 0.72 CHRM2 (0.32) NPSR1CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2222162-A2 SMALL MOLECULE MYRISTATE INHIBITORS OF BCR-ABL AND METHODS OF USE Dana Farber Cancer Institute (US) 2010-09-01 EP disclosed
WO-2009073153-A2 SMALL MOLECULE MYRISTATE INHIBITORS OF BCR-ABL AND METHODS OF USE DANA FARBER CANCER INSTITUTE (US) 2009-06-11 WO disclosed
US-4201784-A ANTITUMOR INSTITUT ORGANICHESKOGO SINTEZA AKADEMII NAUK LATVIISKOI SSR (SU) 1980-05-06 US disclosed