SCHEMBL3401775

SCHEMBL3401775

CC(C)(C)OC(=O)Nc1cc(F)c(F)cc1CO

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CYP17A1 P05093 2/20 0.41
KCNQ4 P56696 3/20 0.40
KCNQ5 Q9NR82 3/20 0.40
RXFP1 Q9HBX9 1/20 0.38
AAK1 Q2M2I8 2/20 0.38
BRAF P15056 1/20 0.36
BRD4 O60885 1/20 0.35
LMNA P02545 1/20 0.35
POLB P06746 1/20 0.35
MTNR1A P48039 1/20 0.35
MTNR1B P49286 1/20 0.35
DPP4 P27487 1/20 0.35
CNR2 P34972 1/20 0.35
DPP8 Q6V1X1 1/20 0.35
DPP9 Q86TI2 1/20 0.35
RORC P51449 1/20 0.35
APLNR P35414 1/20 0.35
BRD9 Q9H8M2 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29071984 0.89 AAK1 (0.47) CYP17A1KCNQ4KCNQ5RXFP1AAK1
SCHEMBL29393326 0.89 AAK1 (0.47) CYP17A1KCNQ4KCNQ5RXFP1AAK1
SCHEMBL3401610 0.87 CYP17A1 (0.40) CYP17A1KCNQ4KCNQ5RXFP1AAK1
SCHEMBL14725520 0.82 CYP17A1 (0.48) CYP17A1KCNQ4KCNQ5RXFP1AAK1
SCHEMBL19501761 0.82 LMNA (0.42) CYP17A1KCNQ4KCNQ5RXFP1AAK1
SCHEMBL29675308 0.80 KDM4A (0.44) LMNA
SCHEMBL22482387 0.80 KDM4A (0.44) LMNA
SCHEMBL3402389 0.80 CA12 (0.38) CYP17A1KCNQ4KCNQ5RXFP1AAK1
SCHEMBL2212401 0.80 CETP (0.42) LMNAPOLBDPP4DPP8DPP9
SCHEMBL22482353 0.80 CYP17A1 (0.43) CYP17A1KCNQ4KCNQ5RXFP1AAK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2250157-B1 NOVEL HETEROCYCLIC COMPOUNDS PANACEA BIOTEC LTD (IN) 2014-11-05 EP disclosed
US-8455479-B2 Heterocyclic compounds PANACEA BIOTEC LIMITED (IN) 2013-06-04 US disclosed
US-20100311732-A1 NOVEL HETEROCYCLIC COMPOUNDS PANACEA BIOTEC PHARMA LIMITED (IN) 2010-12-09 US disclosed
EP-2250157-A1 NOVEL HETEROCYCLIC COMPOUNDS Panacea Biotec Limited (IN) 2010-11-17 EP disclosed
WO-2009093269-A1 NOVEL HETEROCYCLIC COMPOUNDS PANACEA BIOTEC LIMITED (IN) 2009-07-30 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100311732-A1 NOVEL HETEROCYCLIC COMPOUNDS DPP4, DPP3, DPP8 CYP17A1 1100/4885KCNQ4 1813/4885KCNQ5 2394/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.