SCHEMBL3402453

SCHEMBL3402453

COc1ccccc1-c1nc(C)c(C(=O)N2CCN(C(C)C)CC2)s1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 8/20 0.55
CNR1 P21554 1/20 0.48
PARP1 P09874 1/20 0.43
NPC1 O15118 4/20 0.43
RAB9A P51151 3/20 0.43
MAPT P10636 3/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
MEN1 O00255 1/20 0.42
CASP1 P29466 1/20 0.42
HTT P42858 1/20 0.42
KMT2A Q03164 1/20 0.42
ALDH1A1 P00352 3/20 0.42
POLB P06746 1/20 0.42
HPGD P15428 1/20 0.42
KDM4E B2RXH2 1/20 0.42
TSHR P16473 1/20 0.42
HSD17B10 Q99714 1/20 0.42
LMNA P02545 2/20 0.41
CES2 O00748 1/20 0.41
TDP1 Q9NUW8 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3405280 0.89 HTR2C (0.53) HTR2CCNR1PARP1MAPTMEN1
SCHEMBL3402656 0.88 HTR2C (0.48) HTR2CCNR1PARP1MAPTSMN1; SMN2
SCHEMBL3401691 0.88 HTR2C (0.45) HTR2CCNR1MAPTSMN1; SMN2HTT
SCHEMBL3402439 0.88 HTR2C (0.46) HTR2CCNR1PARP1NPC1RAB9A
SCHEMBL13309912 0.87 HTR2C (0.59) HTR2CCNR1PARP1MAPTSMN1; SMN2
SCHEMBL3397009 0.86 HTR2C (0.45) HTR2CCNR1PARP1MAPTALDH1A1
SCHEMBL3399364 0.86 HTR2C (0.45) HTR2CCNR1MAPTMEN1KMT2A
SCHEMBL3400042 0.86 HTR2C (0.58) HTR2CCNR1PARP1MAPTSMN1; SMN2
SCHEMBL3401442 0.85 HTR2C (0.46) HTR2CCNR1PARP1ALDH1A1HPGD
SCHEMBL3404790 0.85 HTR2C (0.57) HTR2CCNR1PARP1NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7728009-B1 Thiazole amides, imidazole amides and related analogues NEUROGEN CORPORATION (US) 2010-06-01 US disclosed
US-7728009-B1 Thiazole amides, imidazole amides and related analogues NEUROGEN CORPORATION (US) 2010-06-01 US disclosed
US-7728009-B1 Thiazole amides, imidazole amides and related analogues NEUROGEN CORPORATION (US) 2010-06-01 US disclosed