SCHEMBL3401442

SCHEMBL3401442

COc1ccc(-c2nc(C)c(C(=O)N3CCN(C(C)C)CC3)s2)c(OC)c1OC

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 7/20 0.46
CNR1 P21554 1/20 0.42
HRH3 Q9Y5N1 2/20 0.40
CFTR P13569 1/20 0.39
HDAC3 O15379 1/20 0.39
HDAC4 P56524 1/20 0.39
HDAC1 Q13547 1/20 0.39
HDAC7 Q8WUI4 1/20 0.39
HDAC2 Q92769 1/20 0.39
HDAC10 Q969S8 1/20 0.39
HDAC11 Q96DB2 1/20 0.39
HDAC8 Q9BY41 1/20 0.39
HDAC6 Q9UBN7 1/20 0.39
HDAC9 Q9UKV0 1/20 0.39
HDAC5 Q9UQL6 1/20 0.39
CYP2C19 P33261 1/20 0.39
SLC6A2 P23975 1/20 0.38
SLC6A4 P31645 1/20 0.38
SLC6A3 Q01959 1/20 0.38
CES2 O00748 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14546080 0.92 HTR2C (0.45) HTR2CCNR1HRH3CFTRCYP2C19
SCHEMBL3402439 0.86 HTR2C (0.46) HTR2CCNR1HRH3CFTRSLC6A2
SCHEMBL3402453 0.85 HTR2C (0.55) HTR2CCNR1HRH3CES2ALDH1A1
SCHEMBL3397009 0.84 HTR2C (0.45) HTR2CCNR1HRH3CFTRSLC6A2
SCHEMBL3401691 0.84 HTR2C (0.45) HTR2CCNR1HRH3CFTRSLC6A2
SCHEMBL3399364 0.84 HTR2C (0.45) HTR2CCNR1HRH3CFTRHDAC1
SCHEMBL3402221 0.83 CNR1 (0.46) HTR2CCNR1HRH3CFTRALDH1A1
SCHEMBL3400850 0.83 HTR2C (0.45) HTR2CHRH3ALDH1A1HPGD
SCHEMBL3404564 0.82 CFTR (0.52) HTR2CCNR1CFTRHDAC6ALDH1A1
SCHEMBL3404031 0.82 HTR2C (0.47) HTR2CCNR1HRH3SLC6A2SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7728009-B1 Thiazole amides, imidazole amides and related analogues NEUROGEN CORPORATION (US) 2010-06-01 US disclosed
US-7728009-B1 Thiazole amides, imidazole amides and related analogues NEUROGEN CORPORATION (US) 2010-06-01 US disclosed
US-7728009-B1 Thiazole amides, imidazole amides and related analogues NEUROGEN CORPORATION (US) 2010-06-01 US disclosed