Nicametate

Nicametate

SCHEMBL34040

CCN(CC)CCOC(=O)c1cccnc1

nearest known ligand 0.68

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 2/20 0.68
LMNA P02545 6/20 0.64
TSHR P16473 3/20 0.59
CYP2D6 P10635 1/20 0.57
MAOA P21397 1/20 0.57
HTR3A P46098 1/20 0.57
HRH3 Q9Y5N1 1/20 0.57
KMT2A Q03164 4/20 0.56
MEN1 O00255 2/20 0.56
SMN1; SMN2 Q16637 1/20 0.56
BLM P54132 1/20 0.56
NPSR1 Q6W5P4 1/20 0.56
SCN1A P35498 1/20 0.55
SCN2A Q99250 1/20 0.55
SCN3A Q9NY46 1/20 0.55
ALDH1A1 P00352 3/20 0.54
MAPT P10636 2/20 0.54
HPGD P15428 1/20 0.54
TDP1 Q9NUW8 1/20 0.54
CYP1A2 P05177 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Nicametate SCHEMBL5060940 1.00 L3MBTL1 (0.68) L3MBTL1LMNATSHRCYP2D6MAOA
Nicametate SCHEMBL28346401 0.96 L3MBTL1 (0.63) L3MBTL1LMNATSHRCYP2D6MAOA
Nicametate SCHEMBL194781 0.87 KDM4E (0.56) L3MBTL1LMNATSHRCYP2D6MAOA
SCHEMBL3079077 0.86 MAPT (0.62) LMNATSHRCYP2D6MAOAHTR3A
Procaine SCHEMBL9312338 0.86 CYP2D6 (0.69) L3MBTL1LMNATSHRCYP2D6MAOA
SCHEMBL9717097 0.85 L3MBTL1 (0.67) L3MBTL1LMNAKMT2AMEN1ALDH1A1
Procaine SCHEMBL9312532 0.85 BLM (0.70) L3MBTL1LMNATSHRCYP2D6MAOA
SCHEMBL382067 0.83 L3MBTL1 (0.82) L3MBTL1LMNATSHRKMT2AMEN1
SCHEMBL25009812 0.83 L3MBTL1 (0.76) L3MBTL1LMNACYP2D6KMT2AMEN1
SCHEMBL30556174 0.83 L3MBTL1 (0.76) L3MBTL1LMNACYP2D6KMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 2484 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4525921-A1 PEPTIDE-IONIC LIQUID CONJUGATE FOR THE PREVENTION AND/OR TREATMENT OF SKIN DISORDERS Universidade Do Porto (PT) 2025-03-26 EP claimed
CN-119438596-A Quick detection method for bacterial drug resistance by combining short-time antibiotic stimulated bacterial metabolism fingerprint spectrum with machine learning 复旦大学 2025-02-14 CN claimed
EP-3607084-B1 A METHOD FOR TESTING ANTIMICROBIAL SUSCEPTIBILITY UNIV WESTERN AUSTRALIA (AU) 2024-05-01 EP claimed
CN-117887673-A Shiga toxin-producing escherichia coli bacteriophage and application thereof in elimination of drug-resistant bacteria 青岛农业大学 2024-04-16 CN claimed
US-11959122-B2 Method for assessing microbial drug resistance multi-level risks of antibiotic residues in water environment Nanjing Institute Of Environmental Sciences, Mee (CN) 2024-04-16 US claimed
WO-2023248196-A1 PEPTIDE-IONIC LIQUID CONJUGATE FOR THE PREVENTION AND/OR TREATMENT OF SKIN DISORDERS UNIVERSIDADE DO PORTO (PT) 2023-12-28 WO claimed
US-20230392183-A1 METHOD FOR ASSESSING MICROBIAL DRUG RESISTANCE MULTI-LEVEL RISKS OF ANTIBIOTIC RESIDUES IN WATER ENVIRONMENT Nanjing Institute Of Environmental Sciences, Mee (CN) 2023-12-07 US claimed
WO-2023183932-A2 MONOBODIES BINDING TO INTERCELLULAR ADHESION MOLECULE 2 (ICAM-2) NEW YORK UNIVERSITY (US) 2023-09-28 WO claimed
CN-115062933-B Multi-level risk assessment method for microbial drug resistance of antibiotic residues in water environment 生态环境部南京环境科学研究所 2023-04-18 CN claimed
CN-115505628-A Combined drug susceptibility test method for rapidly detecting synergistic effect of aztreonam and ceftazidime-abamectin 刘周 2022-12-23 CN claimed
EP-1385501-A2 PROBUCOL MONOESTERS AND THEIR USE TO INCREASE PLASMA HDL CHOLESTEROL LEVELS AND IMPROVE HDL FUNCTIONALITY Atherogenics, Inc. (US) 2004-02-04 EP claimed
WO-2003097714-A1 FAT BINDING USING INTER-POLYMER COMPLEX OF GLUCOSAMINE AND POLYACRYLIC ACID RANBAXY LABORATORIES LIMITED (IN) 2003-11-27 WO claimed
US-20030162824-A1 Methods of treating or preventing a cardiovascular condition using a cyclooxygenase-1 inhibitor PHARMACIA CORPORATION 2003-08-28 US claimed
WO-2002087556-A9 PROBUCOL MONOESTERS AND THEIR USE TO INCREASE PLASMA HDL CHOLESTEROL LEVELS AND IMPROVE HDL FUNCTIONALITY ATHEROGENICS INC (US) 2003-03-20 WO claimed
WO-2002087556-A2 PROBUCOL MONOESTERS AND THEIR USE TO INCREASE PLASMA HDL CHOLESTEROL LEVELS AND IMPROVE HDL FUNCTIONALITY ATHEROGENICS, INC. (US) 2002-11-07 WO claimed
CN-1294519-A Pharmaceutical composition containing a compound having an activity of promoting the absorption of an active ingredient INPHARMA SA (CH) 2001-05-09 CN claimed
EP-1073470-A1 PHARMACEUTICAL COMPOSITIONS CONTAINING COMPOUNDS WITH ACTIVITY FOR THE ENHANCEMENT OF ABSORPTION OF ACTIVE INGREDIENTS INPHARMA S.A. (CH) 2001-02-07 EP claimed
WO-2000048636-A1 PHARMACEUTICAL COMPOSITIONS CONTAINING COMPOUNDS WITH ACTIVITY FOR THE ENHANCEMENT OF ABSORPTION OF ACTIVE INGREDIENTS INPHARMA S.A. (CH) 2000-08-24 WO claimed
US-5938791-A Device for detecting margin of information recording and reproducing apparatus SONY CORPORATION (JP) 1999-08-17 US claimed
EP-0007109-A1 Apparatus for metering a solution of chemicals to a stream of liquid LANG APPARATEBAU GMBH (DE) 1980-01-23 EP claimed