SCHEMBL3405145

SCHEMBL3405145

Cc1ccc(-c2nc(C)c(C(=O)NCCC3CCCN3C)s2)cc1C

nearest known ligand 0.52

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CHRM4 P08173 4/20 0.52
ACKR3 P25106 2/20 0.52
CHRM3 P20309 1/20 0.45
PPARA Q07869 5/20 0.43
NPC1 O15118 1/20 0.43
HPGD P15428 1/20 0.43
BTK Q06187 1/20 0.42
BRAF P15056 1/20 0.42
PPARD Q03181 3/20 0.42
PPARG P37231 2/20 0.42
LCK P06239 1/20 0.42
SCD O00767 1/20 0.42
POLR1A O95602 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3405722 0.92 CHRM4 (0.50) CHRM4ACKR3CHRM3PPARANPC1
SCHEMBL3400749 0.90 CHRM4 (0.49) CHRM4ACKR3PPARABTKPPARD
SCHEMBL3402461 0.89 CHRM4 (0.55) CHRM4ACKR3CHRM3PPARAPPARD
SCHEMBL13309884 0.89 CHRM4 (0.51) CHRM4ACKR3CHRM3PPARAPPARD
SCHEMBL3405362 0.89 ACKR3 (0.55) CHRM4ACKR3PPARANPC1HPGD
SCHEMBL3399661 0.88 CHRM4 (0.53) CHRM4ACKR3CHRM3PPARAPPARD
SCHEMBL3405398 0.87 ACKR3 (0.55) CHRM4ACKR3PPARANPC1HPGD
SCHEMBL3402603 0.87 TLR9 (0.53) CHRM4ACKR3PPARAPPARD
SCHEMBL3403412 0.87 CHRM4 (0.49) CHRM4ACKR3CHRM3PPARABTK
SCHEMBL3401785 0.86 ACKR3 (0.54) CHRM4ACKR3CHRM3PPARANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7728009-B1 Thiazole amides, imidazole amides and related analogues NEUROGEN CORPORATION (US) 2010-06-01 US disclosed
US-7728009-B1 Thiazole amides, imidazole amides and related analogues NEUROGEN CORPORATION (US) 2010-06-01 US disclosed
US-7728009-B1 Thiazole amides, imidazole amides and related analogues NEUROGEN CORPORATION (US) 2010-06-01 US disclosed