SCHEMBL3405362

SCHEMBL3405362

Cc1nc(-c2ccc3ccccc3c2)sc1C(=O)NCCC1CCCN1C

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACKR3 P25106 2/20 0.55
CHRM4 P08173 4/20 0.54
POLR1A O95602 1/20 0.48
NPC1 O15118 1/20 0.46
HPGD P15428 1/20 0.46
BTK Q06187 1/20 0.45
PPARA Q07869 4/20 0.44
PPARD Q03181 3/20 0.44
CHRNB1 P11230 1/20 0.43
CHRNB2 P17787 1/20 0.43
CHRNB4 P30926 1/20 0.43
CHRNA3 P32297 1/20 0.43
CHRNB3 Q05901 1/20 0.43
BRAF P15056 1/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
PPARG P37231 1/20 0.43
ACP1 P24666 1/20 0.43
ALDH1A1 P00352 1/20 0.43
GAA P10253 1/20 0.43
MAPT P10636 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3403412 0.91 CHRM4 (0.49) ACKR3CHRM4BTKPPARAPPARD
SCHEMBL3405442 0.89 ACKR3 (0.59) ACKR3CHRM4NPC1HPGDBTK
SCHEMBL3405145 0.89 CHRM4 (0.52) ACKR3CHRM4POLR1ANPC1HPGD
SCHEMBL3400075 0.88 ACKR3 (0.54) ACKR3CHRM4NPC1HPGDBTK
SCHEMBL3402461 0.87 CHRM4 (0.55) ACKR3CHRM4PPARAPPARDSMN1; SMN2
SCHEMBL13309884 0.87 CHRM4 (0.51) ACKR3CHRM4PPARAPPARDPPARG
SCHEMBL3401785 0.87 ACKR3 (0.54) ACKR3CHRM4NPC1HPGDPPARA
SCHEMBL3405722 0.86 CHRM4 (0.50) ACKR3CHRM4NPC1HPGDBTK
SCHEMBL3403460 0.86 CHRM4 (0.54) ACKR3CHRM4NPC1HPGDPPARA
SCHEMBL3403598 0.86 ACKR3 (0.53) ACKR3CHRM4PPARAPPARDPPARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7728009-B1 Thiazole amides, imidazole amides and related analogues NEUROGEN CORPORATION (US) 2010-06-01 US disclosed
US-7728009-B1 Thiazole amides, imidazole amides and related analogues NEUROGEN CORPORATION (US) 2010-06-01 US disclosed
US-7728009-B1 Thiazole amides, imidazole amides and related analogues NEUROGEN CORPORATION (US) 2010-06-01 US disclosed
WO-2006089076-A9 THIAZOLE AMIDES, IMIDAZOLE AMIDES AND RELATED ANALOGUES NEUROGEN CORP (US) 2007-04-26 WO disclosed