SCHEMBL3405754

SCHEMBL3405754

CCOc1cccc(-c2nc(C)c(C(=O)NCCCCN3CCCC3)s2)c1

nearest known ligand 0.47

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.47
TSHR P16473 1/20 0.47
MAPT P10636 2/20 0.46
NPC1 O15118 1/20 0.46
HPGD P15428 1/20 0.46
HTR1A P08908 3/20 0.45
HTR2A P28223 3/20 0.45
DRD3 P35462 3/20 0.45
HRH3 Q9Y5N1 6/20 0.45
SMYD2 Q9NRG4 2/20 0.45
HTR2C P28335 1/20 0.44
GAA P10253 1/20 0.44
GLA P06280 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
AVPR1B P47901 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3429158 0.94 GLA (0.51) ALDH1A1MAPTNPC1HPGDGAA
SCHEMBL3429141 0.93 GLA (0.50) ALDH1A1TSHRMAPTNPC1HPGD
SCHEMBL3404144 0.88 PPARA (0.47) MAPTNPC1HPGDHTR1AHTR2A
SCHEMBL3402374 0.87 SMYD2 (0.49) NPC1HPGDHTR1AHTR2ADRD3
SCHEMBL3401173 0.85 MAPT (0.50) MAPTNPC1HPGDHTR1AHTR2A
SCHEMBL3405815 0.85 MAPT (0.52) MAPTNPC1HPGDSMYD2
SCHEMBL3398623 0.85 SMYD2 (0.52) MAPTNPC1HPGDHTR1AHTR2A
SCHEMBL3403357 0.84 DRD3 (0.49) TSHRNPC1HPGDHTR1AHTR2A
SCHEMBL3400521 0.84 GAA (0.45) ALDH1A1MAPTNPC1HPGDHTR1A
SCHEMBL3399687 0.84 CHRM4 (0.52) ALDH1A1MAPTNPC1HPGDHRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7728009-B1 Thiazole amides, imidazole amides and related analogues NEUROGEN CORPORATION (US) 2010-06-01 US disclosed
US-7728009-B1 Thiazole amides, imidazole amides and related analogues NEUROGEN CORPORATION (US) 2010-06-01 US disclosed
US-7728009-B1 Thiazole amides, imidazole amides and related analogues NEUROGEN CORPORATION (US) 2010-06-01 US disclosed
WO-2006089076-A9 THIAZOLE AMIDES, IMIDAZOLE AMIDES AND RELATED ANALOGUES NEUROGEN CORP (US) 2007-04-26 WO disclosed