SCHEMBL3400521

SCHEMBL3400521

CSc1cccc(-c2nc(C)c(C(=O)NCCCCN3CCCC3)s2)c1

nearest known ligand 0.45

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.45
NPC1 O15118 1/20 0.45
HPGD P15428 1/20 0.45
SMYD2 Q9NRG4 2/20 0.45
CHRM4 P08173 2/20 0.43
DRD3 P35462 3/20 0.43
HTR1A P08908 2/20 0.43
HTR2A P28223 2/20 0.43
SMN1; SMN2 Q16637 2/20 0.42
HRH3 Q9Y5N1 2/20 0.42
ALDH1A1 P00352 1/20 0.42
MAPT P10636 1/20 0.42
TP53 P04637 1/20 0.42
DRD2 P14416 2/20 0.41
HDAC3 O15379 1/20 0.41
HDAC1 Q13547 1/20 0.41
DRD4 P21917 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3402472 0.94 HPGD (0.47) GAANPC1HPGDSMYD2CHRM4
SCHEMBL3405410 0.93 HPGD (0.47) GAANPC1HPGDCHRM4SMN1; SMN2
SCHEMBL3401173 0.87 MAPT (0.50) GAANPC1HPGDSMYD2CHRM4
SCHEMBL3398623 0.86 SMYD2 (0.52) GAANPC1HPGDSMYD2DRD3
SCHEMBL13309646 0.85 HPGD (0.47) GAANPC1HPGDCHRM4SMN1; SMN2
SCHEMBL3403850 0.85 ALDH1A1 (0.57) GAANPC1HPGDSMYD2CHRM4
SCHEMBL3401375 0.85 SMYD2 (0.51) GAANPC1HPGDSMYD2CHRM4
SCHEMBL3402848 0.85 LMNA (0.52) NPC1HRH3MAPTTP53
SCHEMBL3403357 0.84 DRD3 (0.49) GAANPC1HPGDSMYD2CHRM4
SCHEMBL3405754 0.84 ALDH1A1 (0.47) GAANPC1HPGDSMYD2DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7728009-B1 Thiazole amides, imidazole amides and related analogues NEUROGEN CORPORATION (US) 2010-06-01 US disclosed
US-7728009-B1 Thiazole amides, imidazole amides and related analogues NEUROGEN CORPORATION (US) 2010-06-01 US disclosed
US-7728009-B1 Thiazole amides, imidazole amides and related analogues NEUROGEN CORPORATION (US) 2010-06-01 US disclosed
WO-2006089076-A9 THIAZOLE AMIDES, IMIDAZOLE AMIDES AND RELATED ANALOGUES NEUROGEN CORP (US) 2007-04-26 WO disclosed