SCHEMBL3406869

SCHEMBL3406869

CCN(Cc1ccc(Cl)cc1Cl)c1cccc(-c2cccc(C(=O)NCCO)c2)n1.O=C(NCCO)c1cccc(-c2cccc(NCc3ccc(Cl)cc3Cl)n2)c1

nearest known ligand 0.46

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 11/20 0.46
GPR52 Q9Y2T5 1/20 0.40
PTGDR Q13258 1/20 0.40
FYN P06241 1/20 0.39
ALOX5 P09917 1/20 0.38
EPHX2 P34913 1/20 0.38
MAP4K4 O95819 1/20 0.38
LMNA P02545 1/20 0.37
MAPK1 P28482 1/20 0.37
NLRP1 Q9C000 1/20 0.37
GPR39 O43194 1/20 0.37
GCG P01275 1/20 0.37
GCGR P47871 1/20 0.37
KDR P35968 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL960678 0.93 CNR1 (0.50) CNR1GPR52PTGDRFYNALOX5
SCHEMBL958112 0.88 GPR52 (0.48) CNR1GPR52PTGDRFYNEPHX2
SCHEMBL960125 0.75 PTGDR (0.57) CNR1PTGDRLMNAGPR39
SCHEMBL961208 0.74 CNR1 (0.49) CNR1PTGDRLMNAGPR39
SCHEMBL959317 0.74 GPR52 (0.52) CNR1GPR52FYNMAP4K4KDR
SCHEMBL1513331 0.69 FYN (0.48) GPR52PTGDRFYNMAP4K4LMNA
SCHEMBL960460 0.68 FYN (0.50) GPR52FYNMAP4K4
SCHEMBL1513123 0.67 FYN (0.46) GPR52PTGDRFYNMAP4K4
SCHEMBL1513274 0.66 FYN (0.49) GPR52PTGDRFYNEPHX2MAP4K4
SCHEMBL1513288 0.65 FYN (0.43) CNR1GPR52PTGDRFYNEPHX2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2253618-A1 COMPOUND HAVING 6-MEMBERED AROMATIC RING Takeda Pharmaceutical Company Limited (JP) 2010-11-24 EP disclosed