SCHEMBL3406916

SCHEMBL3406916

CNC1(C#N)CCC(Cc2ccccc2)(CN(C)C)CC1

nearest known ligand 0.64

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
OPRL1 P41146 6/20 0.64
OPRM1 P35372 4/20 0.64
KDM1A O60341 1/20 0.39
CTSS P25774 5/20 0.38
CTSK P43235 5/20 0.38
CTSL P07711 3/20 0.36
SMN1; SMN2 Q16637 1/20 0.35
CTSB P07858 4/20 0.35
OPRK1 P41145 1/20 0.35
SLC6A2 P23975 1/20 0.34
SLC6A4 P31645 1/20 0.34
SLC6A3 Q01959 1/20 0.34
MAOB P27338 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6138260 0.82 OPRL1 (0.78) OPRL1OPRM1KDM1AOPRK1SLC6A2
SCHEMBL3409102 0.82 OPRL1 (0.61) OPRL1OPRM1KDM1ACTSSCTSK
SCHEMBL3411324 0.78 OPRL1 (1.00) OPRL1OPRM1KDM1AOPRK1SLC6A2
SCHEMBL4348241 0.73 OPRL1 (0.60) OPRL1OPRM1KDM1AOPRK1SLC6A2
SCHEMBL3407538 0.73 OPRM1 (0.42) OPRL1OPRM1CTSSCTSKCTSL
SCHEMBL3408991 0.73 OPRL1 (1.00) OPRL1OPRM1OPRK1
SCHEMBL3413567 0.71 OPRL1 (0.61) OPRL1OPRM1KDM1AOPRK1SLC6A2
SCHEMBL3413008 0.71 OPRL1 (0.61) OPRL1OPRM1OPRK1
SCHEMBL4352487 0.70 OPRL1 (0.60) OPRL1OPRM1KDM1AOPRK1SLC6A2
SCHEMBL5242605 0.69 OPRM1 (0.60) OPRL1OPRM1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2502907-B1 Substituted 4-aminocyclohexane derivatives GRUENENTHAL GMBH (DE) 2018-08-29 EP disclosed
EP-2518052-B1 Substituted 4-aminocyclohexane derivatives GRUENENTHAL GMBH (DE) 2017-12-20 EP disclosed
EP-2260021-B1 SUBSTITUTED 4-AMINOCYCLOHEXANE DERIVATIVES GRUENENTHAL GMBH (DE) 2014-04-23 EP disclosed
EP-2518052-A1 Substituted 4-aminocyclohexane derivatives Grünenthal GmbH (DE) 2012-10-31 EP disclosed
EP-2502907-A1 Substituted 4-aminocyclohexane derivatives Grünenthal GmbH (DE) 2012-09-26 EP disclosed
EP-2260021-A1 SUBSTITUTED 4-AMINOCYCLOHEXANE DERIVATIVES Grünenthal GmbH (DE) 2010-12-15 EP disclosed
WO-2009118168-A1 SUBSTITUTED 4-AMINOCYCLOHEXANE DERIVATIVES Grünenthal GmbH (DE) 2009-10-01 WO disclosed