SCHEMBL3407170

SCHEMBL3407170

CCC(=O)C(C)(N)c1cccc(Br)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.44
CYP2C19 P33261 1/20 0.44
GAA P10253 1/20 0.44
SMN1; SMN2 Q16637 2/20 0.43
PARP1 P09874 1/20 0.43
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
CA5A P35218 1/20 0.41
CA9 Q16790 1/20 0.41
RIPK1 Q13546 1/20 0.40
TP53BP1 Q12888 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
KIF11 P52732 1/20 0.38
ALDH1A1 P00352 2/20 0.38
RAB9A P51151 2/20 0.38
NPC1 O15118 1/20 0.38
LMNA P02545 1/20 0.38
HTT P42858 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2171798 0.81 CYP1A2 (0.59) CYP1A2CYP2C19GAASMN1; SMN2PARP1
Hydrochloric Acid SCHEMBL362914 0.80 CYP1A2 (0.58) CYP1A2CYP2C19GAASMN1; SMN2PARP1
Hydrochloric Acid SCHEMBL1173192 0.80 CYP1A2 (0.58) CYP1A2CYP2C19GAASMN1; SMN2PARP1
SCHEMBL1173430 0.77 KMT2A (0.43) CYP1A2CYP2C19GAASMN1; SMN2PARP1
SCHEMBL245200 0.77 KMT2A (0.43) CYP1A2CYP2C19GAASMN1; SMN2PARP1
SCHEMBL27498317 0.77 MEN1 (0.53) GAASMN1; SMN2PARP1MEN1KMT2A
SCHEMBL3186037 0.74 CA1 (0.41) CYP1A2CYP2C19GAASMN1; SMN2PARP1
SCHEMBL21981930 0.74 CYP2C19 (0.47) CYP1A2CYP2C19GAASMN1; SMN2PARP1
SCHEMBL21981929 0.74 CYP2C19 (0.47) CYP1A2CYP2C19GAASMN1; SMN2PARP1
SCHEMBL875111 0.74 CA1 (0.43) CYP1A2CYP2C19GAASMN1; SMN2PARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012000933-A1 3-AMINO-5,6-DIHYDRO-1H-PYRAZIN-2-ONE DERIVATIVES USEFUL FOR THE TREATEMENT OF ALZHEIMER'S DISEASE AND OTHER FORMS OF DEMENTIA JANSSEN PHARMACEUTICA NV (BE) 2012-01-05 WO disclosed