SCHEMBL3408635

SCHEMBL3408635

CC(C)(C)OC(=O)ON1CC2=C(C1)CN(c1ncc(C(=O)NCCCc3ccccc3)s1)C2

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 6/20 0.50
NPC1 O15118 4/20 0.42
RAB9A P51151 3/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
USP2 O75604 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
HDAC3 O15379 2/20 0.40
HDAC4 P56524 2/20 0.40
HDAC1 Q13547 2/20 0.40
HDAC7 Q8WUI4 2/20 0.40
HDAC2 Q92769 2/20 0.40
HDAC10 Q969S8 2/20 0.40
HDAC11 Q96DB2 2/20 0.40
HDAC8 Q9BY41 2/20 0.40
HDAC6 Q9UBN7 2/20 0.40
HDAC9 Q9UKV0 2/20 0.40
HDAC5 Q9UQL6 2/20 0.40
SNCA P37840 1/20 0.40
LIPG Q9Y5X9 1/20 0.39
CYP1A2 P05177 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8093604 0.90 NAMPT (0.54) NAMPTNPC1RAB9ASMN1; SMN2USP2
SCHEMBL2298576 0.84 NAMPT (0.61) NAMPTNPC1RAB9ASMN1; SMN2USP2
SCHEMBL3407350 0.83 NAMPT (0.46) NAMPTHDAC3HDAC4HDAC1HDAC7
SCHEMBL2297912 0.80 NAMPT (0.58) NAMPTNPC1RAB9ASMN1; SMN2USP2
SCHEMBL3402356 0.79 SCD (0.38) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL2297342 0.78 SCD (0.55) NAMPT
SCHEMBL2294218 0.76 NAMPT (0.51) NAMPTNPC1RAB9ASMN1; SMN2USP2
SCHEMBL8093277 0.75 NAMPT (0.47) NAMPTNPC1RAB9ASMN1; SMN2USP2
SCHEMBL2295194 0.75 NAMPT (0.47) NAMPTHDAC3HDAC4HDAC1HDAC7
SCHEMBL3404518 0.75 OGA (0.43) HDAC3HDAC4HDAC1HDAC7HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2152711-B1 2 -HETEROARYL- PYRROLO [3, 4-C]PYRROLE DERIVATIVES AND THEIR USE AS SCD INHIBITORS SANOFI AVENTIS (FR) 2010-11-24 EP disclosed
EP-2152711-A1 2 -HETEROARYL- PYRROLO [3, 4-C]PYRROLE DERIVATIVES AND THEIR USE AS SCD INHIBITORS Sanofi-Aventis (FR) 2010-02-17 EP disclosed
WO-2008135141-A1 2 -HETEROARYL- PYRROLO [3, 4-C] PYRROLE DERIVATIVES AND THEIR USE AS SCD INHIBITORS SANOFI-AVENTIS (FR) 2008-11-13 WO disclosed