SCHEMBL3408718

SCHEMBL3408718

O=C(O)CNc1nc2c(s1)C=CN(c1cn(Cc3cc(Cl)c(Cl)c(Cl)c3)nn1)C2

nearest known ligand 0.37

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
EGLN1 Q9GZT9 2/20 0.33
SIGMAR1 Q99720 1/20 0.31
PTGS2 P35354 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2365301 0.86 SIGMAR1 (0.30) SIGMAR1
SCHEMBL2177486 0.69 EGLN1 (0.42) EGLN1
SCHEMBL2176563 0.68 EGLN1 (0.41) EGLN1
SCHEMBL12408994 0.62 EGLN1 (0.40) EGLN1
SCHEMBL1965690 0.61 EGLN1 (0.44) EGLN1
SCHEMBL1971349 0.59 SCD (0.49)
SCHEMBL2177885 0.58 SCD (0.48) SIGMAR1
SCHEMBL1974270 0.58 SCD (0.66)
SCHEMBL1986750 0.58 SCD (0.40) EGLN1
SCHEMBL1986109 0.57 SCD (0.48)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010037225-A1 HETEROAROMATIC COMPOUNDS AS INHIBITORS OF STEAROYL-COENZYME A DELTA-9 DESATURASE MERCK FROSST CANADA LTD. (CA) 2010-04-08 WO disclosed