SCHEMBL3411435

SCHEMBL3411435

FC(F)(c1ccc2ncccc2c1)c1cnc2ccc(Cl)nn12

nearest known ligand 0.53

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MET P08581 16/20 0.53
PDE3A Q14432 2/20 0.48
NQO2 P16083 1/20 0.48
PDE3B Q13370 1/20 0.48
PIP4K2C Q8TBX8 1/20 0.48
DYRK1A Q13627 3/20 0.45
DYRK2 Q92630 3/20 0.45
DYRK1B Q9Y463 2/20 0.45
CCNA2 P20248 1/20 0.45
CDK2 P24941 1/20 0.45
CDK5 Q00535 1/20 0.45
CDK5R1 Q15078 1/20 0.45
MKNK1 Q9BUB5 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3411011 0.88 MET (0.54) METPDE3ANQO2PDE3BPIP4K2C
SCHEMBL3410453 0.85 MET (0.73) METPDE3ANQO2PDE3BPIP4K2C
SCHEMBL1163158 0.84 MET (0.71) METPDE3ANQO2PDE3BPIP4K2C
SCHEMBL1658513 0.78 MET (0.78) METPDE3ANQO2PDE3BPIP4K2C
SCHEMBL2697690 0.78 MET (0.55) METPDE3ANQO2PDE3BPIP4K2C
SCHEMBL10242462 0.76 MET (0.59) METPDE3ANQO2PDE3BPIP4K2C
SCHEMBL1657584 0.76 MET (0.46) METPDE3APDE3BDYRK1ADYRK2
SCHEMBL1163538 0.74 MET (0.63) METDYRK1ADYRK2DYRK1BCCNA2
SCHEMBL1163412 0.74 MET (0.59) METPDE3ANQO2PDE3BPIP4K2C
SCHEMBL3414008 0.73 MET (0.68) MET

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8822468-B2 3-Methyl-imidazo[1,2-b]pyridazine derivatives NOVARTIS AG (CH) 2014-09-02 US disclosed
EP-2265614-A1 IMIDAZO [1,2-B]PYRIDAZINE DERIVATIVES FOR THE TREATMENT OF C-MET TYROSINE KINASE MEDIATED DISEASE Novartis AG (CH) 2010-12-29 EP disclosed
US-20090264406-A1 3-METHYL-IMIDAZO[1,2-B]PYRIDAZINE DERIVATIVES NOVARTIS AG 2009-10-22 US disclosed
WO-2009106577-A1 IMIDAZO [1,2-B] PYRIDAZINE DERIVATIVES FOR THE TREATMENT OF C-MET TYROSINE KINASE MEDIATED DISEASE NOVARTIS AG (CH) 2009-09-03 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090264406-A1 3-METHYL-IMIDAZO[1,2-B]PYRIDAZINE DERIVATIVES MET, ERBB2, ALK MET 1/4885PDE3A 1289/4885NQO2 4207/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.