SCHEMBL3411657

SCHEMBL3411657

CCOC(=O)C(C)c1c(C(F)(F)F)cc(OC)c(-c2ccccc2)c1CN(CC)C(=O)OCc1ccccc1

nearest known ligand 0.46

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PTGDR2 Q9Y5Y4 17/20 0.46
CYP3A4 P08684 2/20 0.46
CYP2C9 P11712 2/20 0.46
TBXA2R P21731 2/20 0.46
PTGIR P43119 2/20 0.46
PTGDR Q13258 2/20 0.46
APP P05067 1/20 0.36
CETP P11597 1/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3406632 0.81 PTGDR2 (0.51) PTGDR2CYP3A4CYP2C9TBXA2RPTGIR
SCHEMBL3695157 0.80 PTGDR2 (0.47) PTGDR2CYP3A4CYP2C9TBXA2RPTGIR
SCHEMBL3391526 0.79 PTGDR2 (0.58) PTGDR2CYP3A4CYP2C9TBXA2RPTGIR
SCHEMBL3691723 0.78 PTGDR2 (0.53) PTGDR2CYP3A4CYP2C9TBXA2RPTGIR
SCHEMBL151506 0.78 PTGDR2 (0.56) PTGDR2CYP3A4CYP2C9TBXA2RPTGIR
SCHEMBL28785884 0.77 PTGDR2 (0.39) PTGDR2CYP3A4CYP2C9TBXA2RPTGIR
SCHEMBL27986022 0.77 PTGDR2 (0.58) PTGDR2CYP3A4CYP2C9TBXA2RPTGIR
SCHEMBL27821184 0.75 PTGDR2 (0.42) PTGDR2CYP3A4CYP2C9TBXA2RPTGIR
SCHEMBL153470 0.73 PTGDR2 (0.54) PTGDR2CYP3A4CYP2C9TBXA2RPTGIR
SCHEMBL150483 0.72 PTGDR2 (0.72) PTGDR2CYP3A4CYP2C9TBXA2RPTGIR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2257524-A1 N,N-DISUBSTITUTED AMINOALKYLBIPHENYL ANTAGONISTS OF PROSTAGLANDIN D2 RECEPTORS Amira Pharmaceuticals, Inc. (US) 2010-12-08 EP disclosed
WO-2009099902-A1 N,N-DISUBSTITUTED AMINOALKYLBIPHENYL ANTAGONISTS OF PROSTAGLANDIN D2 RECEPTORS AMIRA PHARMACEUTICALS, INC. (US) 2009-08-13 WO disclosed