SCHEMBL3412166

SCHEMBL3412166

C=CCC(=O)c1ccc(Br)cc1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 3/20 0.57
HDAC1 Q13547 2/20 0.53
HDAC8 Q9BY41 2/20 0.53
HDAC3 O15379 1/20 0.53
HDAC4 P56524 1/20 0.53
HDAC7 Q8WUI4 1/20 0.53
HDAC2 Q92769 1/20 0.53
HDAC10 Q969S8 1/20 0.53
HDAC11 Q96DB2 1/20 0.53
HDAC6 Q9UBN7 1/20 0.53
HDAC9 Q9UKV0 1/20 0.53
HDAC5 Q9UQL6 1/20 0.53
CES2 O00748 1/20 0.48
CES1 P23141 1/20 0.48
KMT2A Q03164 1/20 0.47
ATM Q13315 1/20 0.47
TGM2 P21980 2/20 0.46
HAO1 Q9UJM8 1/20 0.46
F13A1 P00488 1/20 0.46
LMNA P02545 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1806027 0.81 ALDH5A1 (0.59) LMNACA1CA2NPC1HPGD
SCHEMBL8975154 0.81 HDAC1 (0.61) GSK3BHDAC1HDAC8HDAC3HDAC4
SCHEMBL11738823 0.80 GSK3B (0.53) GSK3BHDAC1HDAC8HDAC3HDAC4
SCHEMBL3415923 0.79 GSK3B (0.57) GSK3BCES2CES1ATMLMNA
SCHEMBL3630757 0.79 TSHR (0.42) KMT2ALMNASMN1; SMN2NPC1HPGD
SCHEMBL14388863 0.79 GSK3B (0.55) GSK3BHDAC1HDAC8HDAC3HDAC4
SCHEMBL27800538 0.79 KDM4E (0.47) KMT2ACA1CA2CYP2C19
SCHEMBL8519584 0.79 NPC1 (0.55) CES2CES1KMT2ATGM2SMN1; SMN2
SCHEMBL6975977 0.79 GSK3B (0.57) GSK3BHDAC1HDAC8HDAC3HDAC4
Water SCHEMBL27991728 0.79 HDAC1 (0.59) GSK3BHDAC1HDAC8HDAC3HDAC4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 15 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1468994-B1 Process for preparing cyclic amine substituted phenyl-alkyl-ketones BASF SE (DE) 2010-11-24 EP claimed
CN-1072662-C Cyclic amine-substituted phenylalkyl ketones and process for their preparation CIBA SC HOLDING AG (CH) 2001-10-10 CN claimed
US-5977357-A Phenyl alkyl ketone substituted by cyclic amine and a process for the preparation thereof CIBA SPECIALTY CHEMICAL CORPORATION (US) 1999-11-02 US claimed
US-5795985-A Phenyl alkyl ketone substituted by cyclic amine and a process for the preparation thereof CIBA SPECIALTY CHEMICALS CORPORATION (US) 1998-08-18 US claimed
CN-1166487-A Cyclic amine-substituted phenylalkyl ketones and process for their preparation CIBA GEIGY AG (CH) 1997-12-03 CN claimed
JP-6321844-A None JP disclosed
CN-1168700-C Cyclic amine substd. phenylalkanone and preparing method thereof ϣ�����⻯ѧ�عɹ�˾ 2004-09-29 CN disclosed
CN-1072662-C Cyclic amine-substituted phenylalkyl ketones and process for their preparation CIBA SC HOLDING AG (CH) 2001-10-10 CN disclosed
CN-1309116-A Cyclic amine substd. phenylalkanone and preparing method thereof CIBA SC HOLDING AG (CH) 2001-08-22 CN disclosed
US-6191182-B1 SUBJECTING P-HALOPHENYL ALKYL KETONE TO AMINOLYSIS WITH CYCLIC SECONDARY AMINE TO FORM CYCLIC AMINE-SUBSTITUTED PHENYL ALKYL KETONE; HALOGINATION AND REACTING WITH AMINE COMPOUND; STEVENS REARRANGEMENT UNDER BASIC CONDITION CIBA SPECIALTY CHEMCIALS CORPORATION 2001-02-20 US disclosed
US-5977357-A Phenyl alkyl ketone substituted by cyclic amine and a process for the preparation thereof CIBA SPECIALTY CHEMICAL CORPORATION (US) 1999-11-02 US disclosed
US-5922898-A Process for preparing biaryl compounds CATALYTICA PHARMACEUTICALS, INC. (US) 1999-07-13 US disclosed
US-5795985-A Phenyl alkyl ketone substituted by cyclic amine and a process for the preparation thereof CIBA SPECIALTY CHEMICALS CORPORATION (US) 1998-08-18 US disclosed
CN-1166487-A Cyclic amine-substituted phenylalkyl ketones and process for their preparation CIBA GEIGY AG (CH) 1997-12-03 CN disclosed
JP-H06321844-A TOLAN DERIVATIVE COMPOUND, LIQUID CRYSTAL MATERIAL AND LIQUID CRYSTAL ELEMENT CONTAINING THE SAME JAPAN CARLIT CO LTD:THE 1994-11-22 JP disclosed