SCHEMBL3416883

SCHEMBL3416883

Cc1nc(C(=O)N2C[C@@H]3C[C@@H]3[C@H]2C(N)=O)c(-c2cccc(F)c2)o1

nearest known ligand 0.40

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 8/20 0.40
HCRTR2 O43614 7/20 0.40
PDE4B Q07343 2/20 0.40
FPR2 P25090 1/20 0.39
GRM5 P41594 5/20 0.36
PIK3CA P42336 1/20 0.36
SLC9A1 P19634 1/20 0.36
MAOA P21397 1/20 0.35
MAOB P27338 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3416884 0.86 FPR2 (0.41) HCRTR1HCRTR2PDE4BFPR2GRM5
SCHEMBL3411921 0.81 HCRTR1 (0.50) HCRTR1HCRTR2
SCHEMBL3415419 0.81 HCRTR1 (0.50) HCRTR1HCRTR2
SCHEMBL3409379 0.81 HCRTR1 (0.50) HCRTR1HCRTR2
SCHEMBL3409382 0.81 HCRTR1 (0.50) HCRTR1HCRTR2
SCHEMBL2926675 0.81 HCRTR1 (0.50) HCRTR1HCRTR2
SCHEMBL2931039 0.78 HCRTR2 (0.39) HCRTR1HCRTR2PDE4BGRM5
SCHEMBL3413130 0.78 HCRTR1 (0.40) HCRTR1HCRTR2PIK3CA
SCHEMBL2931852 0.78 HCRTR1 (0.40) HCRTR1HCRTR2PIK3CA
SCHEMBL2056738 0.78 HCRTR1 (0.43) HCRTR1HCRTR2FPR2GRM5SLC9A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2185512-B1 TRANS-3-AZA-BICYCLO[3.1.0]HEXANE DERIVATIVES ACTELION PHARMACEUTICALS LTD (CH) 2010-12-29 EP disclosed