Miproxifene

Miproxifene

SCHEMBL34173

CC/C(=C(\c1ccc(O)cc1)c1ccc(OCCN(C)C)cc1)c1ccc(C(C)C)cc1

nearest known ligand 0.76

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 14/20 0.76
ESR2 Q92731 7/20 0.76
ESRRG P62508 4/20 0.76
MAPT P10636 3/20 0.76
CYP3A4 P08684 3/20 0.76
ESRRB O95718 3/20 0.76
MEN1 O00255 2/20 0.76
TP53 P04637 2/20 0.76
KMT2A Q03164 2/20 0.76
PGR P06401 2/20 0.76
KDM4E B2RXH2 1/20 0.76
ALDH1A1 P00352 1/20 0.76
LMNA P02545 1/20 0.76
HIF1A Q16665 1/20 0.76
NPSR1 Q6W5P4 1/20 0.76
PLD2 O14939 1/20 0.76
PLD1 Q13393 1/20 0.76
HDAC6 Q9UBN7 5/20 0.69
CYP1A2 P05177 2/20 0.67
CYP2D6 P10635 2/20 0.67

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Miproxifene SCHEMBL409028 1.00 ESR1 (0.76) ESR1ESR2ESRRGMAPTCYP3A4
Miproxifene SCHEMBL409027 1.00 ESR1 (0.76) ESR1ESR2ESRRGMAPTCYP3A4
Miproxifene SCHEMBL9857626 0.99 ESR1 (0.74) ESR1ESR2ESRRGMAPTCYP3A4
Miproxifene SCHEMBL9857619 0.99 ESR1 (0.74) ESR1ESR2ESRRGMAPTCYP3A4
Miproxifene SCHEMBL9857612 0.99 ESR1 (0.74) ESR1ESR2ESRRGMAPTCYP3A4
Miproxifene SCHEMBL2128564 0.99 ESR1 (0.74) ESR1ESR2ESRRGMAPTCYP3A4
Miproxifene SCHEMBL3781209 0.94 ESR1 (0.69) ESR1ESR2ESRRGMAPTCYP3A4
Miproxifene SCHEMBL430163 0.94 ESR1 (0.69) ESR1ESR2ESRRGMAPTCYP3A4
Miproxifene SCHEMBL3781215 0.94 ESR1 (0.69) ESR1ESR2ESRRGMAPTCYP3A4
SCHEMBL9857240 0.91 ESR1 (0.90) ESR1ESR2ESRRGMAPTCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1300 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12364682-B2 Use of tegaserod in preparation of anti-tumor drug QINGDAO HAIJI BIOMEDICINE CO., LTD. (CN) 2025-07-22 US claimed
US-20250059301-A1 Fusion Protein Construct NORTHWESTERN UNIVERSITY 2025-02-20 US claimed
US-20230338355-A1 NK ANTAGONISTS FOR CONTRACEPTION ACER THERAPEUTICS INC. 2023-10-26 US claimed
WO-2022026901-A2 NK ANTAGONISTS FOR CONTRACEPTION ACER THERAPEUTICS INC. (US) 2022-02-03 WO claimed
US-20210060052-A1 IN SITU METHODS OF INDUCING OF IMMUNE RESPONSE ATOSSA THERAPEUTICS, INC. (US) 2021-03-04 US claimed
EP-3765007-A1 IN SITU METHODS OF INDUCING OF IMMUNE RESPONSE Atossa Therapeutics, Inc. (US) 2021-01-20 EP claimed
US-20210000920-A1 INTRADUCTAL METHODS OF TREATMENT OF BREAST DISORDERS ATOSSA THERAPEUTICS, INC. (US) 2021-01-07 US claimed
EP-3727403-A1 INTRADUCTAL METHODS OF TREATMENT OF BREAST DISORDERS Atossa Therapeutics, Inc. (US) 2020-10-28 EP claimed
US-10561648-B2 Inhibition and treatment of bacterial infections by sex-specific GPER targeting STC.UNM (US) 2020-02-18 US claimed
WO-2019177991-A1 IN SITU METHODS OF INDUCING OF IMMUNE RESPONSE ATOSSA GENETICS, INC. (US) 2019-09-19 WO claimed
JP-2006519264-A 2006-08-24 JP claimed
EP-1599467-A1 NOVEL CYANOPYRIDINE DERIVATIVES USEFUL IN THE TREATMENT OF CANCER AND OTHER DISORDERS Bayer Pharmaceuticals Corporation (US) 2005-11-30 EP claimed
WO-2005110994-A2 SUBSTITUTED PYRAZOLYL UREA DERIVATIVES USEFUL IN THE TREATMENT OF CANCER BAYER PHARMACEUTICALS CORPORATION (US) 2005-11-24 WO claimed
CN-1660437-A Combination of slow released anticancer medication LANJIN BIOLOG ENGINEERING CO L (CN) 2005-08-31 CN claimed
US-20040235829-A1 Novel cyanopyridine derivatives useful in the treatment of cancer and other disorders BAYER HEALTHCARE LLC 2004-11-25 US claimed
EP-1465619-A1 SUPPRESSION OF CARTILAGE DEGRADATION VIA THE ESTROGEN RECEPTOR Nordic Bioscience A/S (DK) 2004-10-13 EP claimed
WO-2004078747-A1 NOVEL CYANOPYRIDINE DERIVATIVES USEFUL IN THE TREATMENT OF CANCER AND OTHER DISORDERS BAYER PHARMACEUTICALS CORPORATION (US) 2004-09-16 WO claimed
WO-2003070253-A1 ESTROGENIC COMPONENT FOR TREATING DECREASED LIBIDO IN WOMEN PANTARHEI BIOSCIENCE B.V. (NL) 2003-08-28 WO claimed
EP-1336602-A1 Nitrate prodrugs able to release nitric oxide in a controlled and selective way and their use for prevention and treatment of inflammatory, ischemic and proliferative diseases Scaramuzzino, Giovanni (IT) 2003-08-20 EP claimed
WO-2003063859-A1 SUPPRESSION OF CARTILAGE DEGRADATION VIA THE ESTROGEN RECEPTOR NORDIC BIOSCIENCE A/S (DK) 2003-08-07 WO claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12364682-B2 Use of tegaserod in preparation of anti-tumor drug STAT3, JAK2, JAK1 ESR1 4633/4885ESR2 4402/4885ESRRG 3780/4885
US-10561648-B2 Inhibition and treatment of bacterial infections by sex-specific GPER targeting GPER1, GPBAR1, ESR1 ESR1 3/4885ESR2 7/4885ESRRG 4/4885
US-20040235829-A1 Novel cyanopyridine derivatives useful in the treatment of cancer and other disorders VHL, HCCS, CDK4 ESR1 4454/4885ESR2 3380/4885ESRRG 4154/4885
US-20250059301-A1 Fusion Protein Construct RPS27A, CD2BP2, JMJD7 ESR1 2980/4885ESR2 3683/4885ESRRG 2696/4885
US-20230338355-A1 NK ANTAGONISTS FOR CONTRACEPTION KLKB1, KLK3, SHBG ESR1 1083/4885ESR2 677/4885ESRRG 310/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.