SCHEMBL3417828

SCHEMBL3417828

Nc1ccc(NCCCCN2CCCN(c3cccc(Cl)c3Cl)CC2)cc1N

nearest known ligand 0.62

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 19/20 0.62
HTR1A P08908 6/20 0.62
HTR2A P28223 4/20 0.62
HTR7 P34969 3/20 0.62
HTR6 P50406 3/20 0.62
DRD3 P35462 12/20 0.56
ADRA1A P35348 7/20 0.56
KCNH2 Q12809 2/20 0.53
HRH4 Q9H3N8 2/20 0.53
DRD4 P21917 5/20 0.51
ADRA1D P25100 2/20 0.51
ADRA1B P35368 2/20 0.51
DRD1 P21728 1/20 0.51
HTR2C P28335 1/20 0.51
HTR2B P41595 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3408350 0.93 DRD2 (0.62) DRD2HTR1AHTR2AHTR7HTR6
SCHEMBL253399 0.82 DRD2 (0.71) DRD2HTR1AHTR2AHTR7HTR6
SCHEMBL252277 0.81 DRD2 (0.67) DRD2HTR1AHTR2AHTR7HTR6
SCHEMBL3418478 0.81 DRD2 (0.72) DRD2HTR1AHTR2AHTR7HTR6
SCHEMBL3402211 0.79 DRD2 (0.73) DRD2HTR1AHTR2AHTR7HTR6
SCHEMBL252996 0.78 DRD2 (0.67) DRD2HTR1AHTR2AHTR7HTR6
SCHEMBL16633520 0.78 DRD2 (0.59) DRD2HTR1AHTR2AHTR7HTR6
SCHEMBL252531 0.78 DRD2 (0.72) DRD2HTR1AHTR2AHTR7HTR6
SCHEMBL252551 0.77 DRD2 (0.71) DRD2HTR1AHTR2AHTR7HTR6
SCHEMBL254909 0.77 DRD2 (0.72) DRD2HTR1AHTR2AHTR7HTR6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012003418-A2 FUNCTIONALLY SELECTIVE LIGANDS OF DOPAMINE D2 RECEPTORS THE UNIVERSITY OF NORTH CAROLINA AT CHAPEL HILL (US) 2012-01-05 WO disclosed