SCHEMBL3418492

SCHEMBL3418492

Nc1ncc(Br)nc1OCCc1c(Cl)ccc(F)c1Cl

nearest known ligand 0.39

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
MET P08581 11/20 0.39
MAP4K3 Q8IVH8 3/20 0.35
JAK2 O60674 2/20 0.35
CCR4 P51679 2/20 0.33
CSF1R P07333 1/20 0.33
EPHB4 P54760 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL488880 0.82 CSF1R (0.38) METMAP4K3JAK2CCR4CSF1R
SCHEMBL1823431 0.79 MET (0.57) METMAP4K3JAK2
SCHEMBL28632433 0.78 CSF1R (0.40) METMAP4K3JAK2CSF1R
SCHEMBL15271269 0.74 MET (0.38) METMAP4K3JAK2EPHB4
SCHEMBL2426505 0.73 MET (0.47) MET
SCHEMBL14812299 0.72 MET (0.54) METMAP4K3JAK2
SCHEMBL1582121 0.72 MET (0.66) METMAP4K3JAK2
SCHEMBL488720 0.72 MET (0.66) METMAP4K3JAK2
SCHEMBL29507219 0.72 CSF1R (0.57) METCCR4CSF1R
SCHEMBL488752 0.72 CSF1R (0.57) METCCR4CSF1R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1784396-B1 PYRAZOLE-SUBSTITUTED AMINOHETEROARYL COMPOUNDS AS PROTEIN KINASE INHIBITORS PFIZER (US) 2010-12-22 EP disclosed