SCHEMBL3419327

SCHEMBL3419327

CC(=NOCc1ccc(C(F)(F)F)cc1)c1ccc(-c2cccc(CC(=O)O)c2)cc1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 8/20 0.63
PPARG P37231 3/20 0.55
PPARA Q07869 3/20 0.55
RXRA P19793 3/20 0.49
NR1H2 P55055 1/20 0.49
NR1H3 Q13133 1/20 0.49
PPARD Q03181 2/20 0.48
PSEN1 P49768 1/20 0.47
PSEN2 P49810 1/20 0.47
APH1B Q8WW43 1/20 0.47
NCSTN Q92542 1/20 0.47
APH1A Q96BI3 1/20 0.47
PSENEN Q9NZ42 1/20 0.47
RXRB P28702 2/20 0.47
RXRG P48443 2/20 0.47
MGLL Q99685 1/20 0.47
NPC1 O15118 1/20 0.47
RAB9A P51151 1/20 0.47
FFAR1 O14842 1/20 0.46
AGXT P21549 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3419326 1.00 S1PR1 (0.63) S1PR1PPARGPPARARXRANR1H2
SCHEMBL3416601 0.92 S1PR1 (0.53) S1PR1PPARGPPARARXRANR1H2
SCHEMBL3416605 0.92 S1PR1 (0.53) S1PR1PPARGPPARARXRANR1H2
SCHEMBL3418738 0.90 S1PR1 (0.62) S1PR1PPARGPPARANPC1RAB9A
SCHEMBL3418743 0.90 S1PR1 (0.62) S1PR1PPARGPPARANPC1RAB9A
SCHEMBL4726495 0.87 S1PR1 (0.66) S1PR1PPARGPPARARXRAPPARD
SCHEMBL3414272 0.86 NPC1 (0.64) S1PR1PPARGPPARANPC1RAB9A
SCHEMBL3414279 0.86 NPC1 (0.64) S1PR1PPARGPPARANPC1RAB9A
SCHEMBL3418794 0.85 PPARG (0.47) S1PR1PPARGPPARARXRANR1H2
SCHEMBL3418793 0.85 PPARG (0.47) S1PR1PPARGPPARARXRANR1H2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7687664-B2 Carboxylic acid derivative, a salt thereof or an ester of them, and medicament comprising it EISAI R&D MANAGEMENT CO., LTD. (JP) 2010-03-30 US disclosed
EP-1394147-A1 CARBOXYLIC ACID DERIVATIVE AND MEDICINE COMPRISING SALT OR ESTER OF THE SAME Eisai Co., Ltd. (JP) 2004-03-03 EP disclosed