SCHEMBL3419476

SCHEMBL3419476

Cc1nc(-c2cccc(F)c2OCc2ccccc2)n(CCc2ccccc2)c(=O)c1-c1cc(-c2nnc(CO)o2)cs1

nearest known ligand 0.54

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
NR1I2 O75469 5/20 0.54
CASR P41180 17/20 0.49
TSHR P16473 2/20 0.35
ALDH1A1 P00352 1/20 0.35
LMNA P02545 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
HIF1A Q16665 1/20 0.35
MAPT P10636 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3418570 0.93 NR1I2 (0.48) NR1I2CASRTSHRALDH1A1LMNA
SCHEMBL3418275 0.92 NR1I2 (0.51) NR1I2CASRTSHRALDH1A1LMNA
SCHEMBL3421089 0.90 NR1I2 (0.50) NR1I2CASRTSHRALDH1A1LMNA
SCHEMBL3418557 0.89 NR1I2 (0.66) NR1I2CASR
SCHEMBL3420836 0.86 NR1I2 (0.50) NR1I2CASRTSHRALDH1A1LMNA
SCHEMBL3349521 0.85 CASR (0.61) NR1I2CASRTSHRALDH1A1LMNA
SCHEMBL3419845 0.84 NR1I2 (0.52) NR1I2CASRTSHRALDH1A1LMNA
SCHEMBL3345165 0.84 CASR (0.56) NR1I2CASRTSHRALDH1A1LMNA
SCHEMBL3415872 0.83 CASR (0.52) NR1I2CASRTSHRALDH1A1LMNA
SCHEMBL3415574 0.83 NR1I2 (0.51) NR1I2CASRTSHRALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010065383-A1 CALCILYTIC COMPOUNDS GLAXOSMITHKLINE LLC (US) 2010-06-10 WO disclosed