SCHEMBL3421652

SCHEMBL3421652

Cn1c(=O)n(CCCCBr)c(=O)c2[nH]cnc21

nearest known ligand 0.75

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 8/20 0.75
ADORA2A P29274 8/20 0.75
PDE4B Q07343 8/20 0.75
PDE4C Q08493 8/20 0.75
PDE4D Q08499 8/20 0.75
ADORA2B P29275 9/20 0.68
ADORA3 P0DMS8 5/20 0.65
CHIT1 Q13231 1/20 0.65
CHIA Q9BZP6 1/20 0.65
CFTR P13569 1/20 0.63
ATAD2 Q6PL18 1/20 0.59
PIK3CD O00329 1/20 0.57
ALPL P05186 1/20 0.57
TMIGD3 P0DMS9 1/20 0.57
ADORA1 P30542 1/20 0.57
CYP2C19 P33261 1/20 0.57
HIF1A Q16665 1/20 0.57
LMNA P02545 1/20 0.56
CYP1A2 P05177 1/20 0.56
MAPT P10636 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21381258 0.87 PDE4A (0.92) PDE4AADORA2APDE4BPDE4CPDE4D
SCHEMBL7458212 0.86 PDE4A (0.89) PDE4AADORA2APDE4BPDE4CPDE4D
SCHEMBL28130992 0.86 PDE4A (0.75) PDE4AADORA2APDE4BPDE4CPDE4D
Iodide SCHEMBL28973314 0.86 PDE4A (0.89) PDE4AADORA2APDE4BPDE4CPDE4D
SCHEMBL27652257 0.86 PDE4A (0.79) PDE4AADORA2APDE4BPDE4CPDE4D
SCHEMBL7109948 0.86 PDE4A (1.00) PDE4AADORA2APDE4BPDE4CPDE4D
SCHEMBL29581286 0.85 PDE4A (0.75) PDE4AADORA2APDE4BPDE4CPDE4D
SCHEMBL9430800 0.85 PDE4A (0.73) PDE4AADORA2APDE4BPDE4CPDE4D
SCHEMBL10854933 0.85 PDE4A (0.73) PDE4AADORA2APDE4BPDE4CPDE4D
SCHEMBL8656750 0.85 PDE4A (0.87) PDE4AADORA2APDE4BPDE4CPDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113816999-B Caffeine-derived azacyclo-carbene-palladium complex and synthesis method and catalytic application thereof 常州大学 2022-08-26 CN disclosed
CN-113816999-A Caffeine-derived azacyclo-carbene-palladium complex and synthesis method and catalytic application thereof 常州大学 2021-12-21 CN disclosed
EP-2159226-B1 ANTIHISTAMINIC AND ANTIALLERGIC AGENT AND A METHOD FOR THE PRODUCTION THEREOF. JOINT STOCK COMPANY OBNINSK CHEMICAL PHARMACEUTICAL COMPANY (RU) 2016-08-31 EP disclosed
EP-2159226-A1 ANTIHISTAMINIC AND ANTIALLERGIC AGENT AND A METHOD FOR THE PRODUCTION THEREOF. Obschestvo S Ogranishennoi Otvetstvennostu "Farmving" (RU) 2010-03-03 EP disclosed