SCHEMBL3423769

SCHEMBL3423769

COc1cc(OC)c(C(=O)O)cc1F

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.55
KDM4E B2RXH2 3/20 0.55
HPGD P15428 2/20 0.55
HTT P42858 2/20 0.55
LMNA P02545 1/20 0.55
MAPK1 P28482 1/20 0.55
RAB9A P51151 1/20 0.55
LCK P06239 1/20 0.53
FYN P06241 1/20 0.53
NPSR1 Q6W5P4 1/20 0.49
HSD17B10 Q99714 2/20 0.49
CYP3A4 P08684 1/20 0.46
PTGS2 P35354 1/20 0.44
CA12 O43570 2/20 0.42
CA1 P00915 2/20 0.42
CA2 P00918 2/20 0.42
CA4 P22748 2/20 0.42
CA6 P23280 2/20 0.42
CA7 P43166 2/20 0.42
CA9 Q16790 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1931203 0.90 ALDH1A1 (0.56) ALDH1A1KDM4EHPGDHTTLMNA
SCHEMBL17700509 0.88 HTT (0.55) ALDH1A1KDM4EHPGDHTTLMNA
SCHEMBL28786089 0.87 LCK (0.73) ALDH1A1KDM4EHPGDHTTLMNA
SCHEMBL12444067 0.85 ALDH1A1 (0.64) ALDH1A1KDM4EHPGDHTTLCK
SCHEMBL19667102 0.85 LCK (0.65) ALDH1A1KDM4EHPGDHTTLMNA
SCHEMBL18713914 0.85 ALDH1A1 (0.51) ALDH1A1KDM4EHPGDHTTLMNA
SCHEMBL7349901 0.85 KDM4E (0.51) ALDH1A1KDM4EHPGDHTTLMNA
SCHEMBL18700941 0.84 HTT (0.55) ALDH1A1KDM4EHPGDHTTLMNA
SCHEMBL31166907 0.84 CYP3A4 (0.50) ALDH1A1KDM4EHPGDHTTLMNA
SCHEMBL7348461 0.84 KDM4E (0.44) ALDH1A1KDM4EHPGDHTTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014203132-A1 SUBSTITUTED BENZOPYRAN COMPOUNDS, COMPOSITIONS AND USES THEREOF OLEMA PHARMACEUTICALS, INC. (US) 2014-12-24 WO disclosed
WO-2014203132-A1 SUBSTITUTED BENZOPYRAN COMPOUNDS, COMPOSITIONS AND USES THEREOF OLEMA PHARMACEUTICALS, INC. (US) 2014-12-24 WO disclosed
US-7759459-B2 Fluorescent assays for protein kinases ALBERT EINSTEIN COLLEGE OF MEDICINE OF YESHIVA UNIVERSITY (US) 2010-07-20 US disclosed
US-7759459-B2 Fluorescent assays for protein kinases ALBERT EINSTEIN COLLEGE OF MEDICINE OF YESHIVA UNIVERSITY (US) 2010-07-20 US disclosed
US-7759459-B2 Fluorescent assays for protein kinases ALBERT EINSTEIN COLLEGE OF MEDICINE OF YESHIVA UNIVERSITY (US) 2010-07-20 US disclosed
US-20050054024-A1 Fluorescent assays for protein kinases NATIONAL INSTITUTES OF HEALTH 2005-03-10 US disclosed
WO-2004062475-A2 FLUORESCENT ASSAYS FOR PROTEIN KINASES ALBERT EINSTEIN COLLEGE OF MEDICINE OF YESHIVA UNIVERSITY (US) 2004-07-29 WO disclosed