SCHEMBL3428177

SCHEMBL3428177

NC(=O)C(SC(F)(F)F)c1ccccc1

nearest known ligand 0.50

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
EPHX1 P07099 12/20 0.50
CTSD P07339 1/20 0.40
CYP2D6 P10635 1/20 0.38
LMNA P02545 1/20 0.38
SRC P12931 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28991897 0.85 SRC (0.45) EPHX1CTSDCYP2D6LMNASRC
SCHEMBL28095496 0.80 TDP1 (0.50) CYP2D6LMNA
SCHEMBL28032290 0.79 EPHX1 (0.39) EPHX1CYP2D6SRC
SCHEMBL28787282 0.78 EPHX1 (0.53) EPHX1CTSDCYP2D6LMNASRC
SCHEMBL1569023 0.75 NPC1 (0.51) EPHX1CTSDCYP2D6LMNA
SCHEMBL6796251 0.73 EPHX1 (0.71) EPHX1LMNA
SCHEMBL1483540 0.72 EPHX1 (0.46) EPHX1CTSDCYP2D6LMNASRC
SCHEMBL19716698 0.72 EPHX1 (0.51) EPHX1CTSDLMNA
Hydrochloric Acid SCHEMBL8413696 0.71 EPHX1 (0.44) EPHX1CTSDCYP2D6LMNASRC
SCHEMBL31130672 0.70 SRC (0.39) CYP2D6LMNASRC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2250162-A2 AMIDE DERIVATIVES AS POSITIVE ALLOSTERIC MODULATORS AND METHODS OF USE THEREOF Abbott Laboratories (US) 2010-11-17 EP disclosed
WO-2009100294-A2 AMIDE DERIVATIVES AS POSITIVE ALLOSTERIC MODULATORS AND METHODS OF USE THEREOF ABBOTT LABORATORIES (US) 2009-08-13 WO disclosed