SCHEMBL3433346

SCHEMBL3433346

CCOC(=O)Cc1ccc(OC)c(-c2ccc(C(F)(F)F)cc2)c1CN(CC)C(=O)NCc1ccccc1O

nearest known ligand 0.45

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PTGDR2 Q9Y5Y4 12/20 0.45
TBXA2R P21731 4/20 0.36
PTGDR Q13258 4/20 0.36
CYP3A4 P08684 2/20 0.36
CYP2C9 P11712 2/20 0.36
PTGIR P43119 2/20 0.36
EPHX2 P34913 1/20 0.34
PPARD Q03181 3/20 0.33
PTGER1 P34995 1/20 0.33
PPARA Q07869 2/20 0.33
PPARG P37231 1/20 0.33
DHFR P00374 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3433468 0.84 PTGDR2 (0.47) PTGDR2TBXA2RPTGDRCYP3A4CYP2C9
SCHEMBL1235425 0.82 PTGDR2 (0.63) PTGDR2TBXA2RPTGDRCYP3A4CYP2C9
SCHEMBL3405517 0.82 PTGDR2 (0.38) PTGDR2TBXA2RPTGDRCYP3A4CYP2C9
SCHEMBL151168 0.79 PTGDR2 (0.71) PTGDR2TBXA2RPTGDRCYP3A4CYP2C9
SCHEMBL3408140 0.79 PTGDR2 (0.59) PTGDR2TBXA2RPTGDRCYP3A4CYP2C9
SCHEMBL3397145 0.79 PPARA (0.39) PPARDPPARAPPARG
SCHEMBL3433349 0.78 PPARA (0.37) PTGDR2EPHX2PPARDPPARAPPARG
SCHEMBL3428160 0.78 PTGDR2 (0.42) PTGDR2TBXA2RPTGDRCYP3A4CYP2C9
SCHEMBL3427454 0.77 PTGDR2 (0.41) PTGDR2TBXA2RPTGDRCYP3A4CYP2C9
SCHEMBL3432155 0.77 PTGDR2 (0.57) PTGDR2TBXA2RPTGDRCYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2257524-A1 N,N-DISUBSTITUTED AMINOALKYLBIPHENYL ANTAGONISTS OF PROSTAGLANDIN D2 RECEPTORS Amira Pharmaceuticals, Inc. (US) 2010-12-08 EP disclosed
WO-2009099902-A1 N,N-DISUBSTITUTED AMINOALKYLBIPHENYL ANTAGONISTS OF PROSTAGLANDIN D2 RECEPTORS AMIRA PHARMACEUTICALS, INC. (US) 2009-08-13 WO disclosed