SCHEMBL3434012

SCHEMBL3434012

Cc1ccc(C(=O)O)c(O)c1NC(=O)c1cc2ccccc2[nH]1

nearest known ligand 0.56

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.56
RAB9A P51151 2/20 0.56
LMNA P02545 1/20 0.56
SMN1; SMN2 Q16637 1/20 0.56
EGFR P00533 7/20 0.50
PIK3CA P42336 7/20 0.50
KDM4E B2RXH2 2/20 0.50
MAPT P10636 1/20 0.50
DAO P14920 1/20 0.50
HPGD P15428 1/20 0.50
SRD5A2 P31213 1/20 0.50
HSD17B10 Q99714 1/20 0.50
CCKAR P32238 1/20 0.50
ALDH1A1 P00352 1/20 0.49
GAA P10253 1/20 0.49
MAPK1 P28482 1/20 0.49
TP53 P04637 1/20 0.48
POLB P06746 1/20 0.48
NHERF1 O14745 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19476086 0.82 NPC1 (0.64) NPC1RAB9ALMNASMN1; SMN2EGFR
SCHEMBL19476095 0.80 NPC1 (0.58) NPC1RAB9ALMNASMN1; SMN2EGFR
SCHEMBL19476161 0.78 NPC1 (0.62) NPC1RAB9ALMNASMN1; SMN2EGFR
SCHEMBL19476092 0.76 NPC1 (0.59) NPC1RAB9ALMNASMN1; SMN2EGFR
SCHEMBL13701154 0.76 NHERF1 (0.74) NPC1RAB9ALMNASMN1; SMN2CCKAR
SCHEMBL29630891 0.75 NPC1 (0.49) NPC1RAB9ALMNASMN1; SMN2KDM4E
SCHEMBL1308155 0.75 NPC1 (0.58) NPC1RAB9ALMNASMN1; SMN2EGFR
SCHEMBL19476162 0.74 NPC1 (0.64) NPC1RAB9ALMNASMN1; SMN2EGFR
SCHEMBL7208136 0.73 NPC1 (1.00) NPC1RAB9ALMNASMN1; SMN2EGFR
SCHEMBL29475123 0.73 NPC1 (1.00) NPC1RAB9ALMNASMN1; SMN2EGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2247600-A2 BENZOXAZOLE CARBOXAMIDE INHIBITORS OF POLY(ADP-RIBOSE)POLYMERASE (PARP) Lead Therapeutics, Inc. (US) 2010-11-10 EP disclosed
WO-2009099736-A2 BENZOXAZOLE CARBOXAMIDE INHIBITORS OF POLY(ADP-RIBOSE)POLYMERASE (PARP) LEAD THERAPEUTICS, INC. (US) 2009-08-13 WO disclosed