SCHEMBL3435652

SCHEMBL3435652

CCCc1ccc(-n2c(Br)nnc2SCC(=O)Nc2ccc(C(=O)O)cc2Cl)c2ccccc12

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC22A12 Q96S37 6/20 0.48
CYP2C9 P11712 2/20 0.43
CYP2C19 P33261 2/20 0.43
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2D6 P10635 1/20 0.43
SLC22A11 Q9NSA0 1/20 0.43
KMT2A Q03164 3/20 0.43
MEN1 O00255 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
GAA P10253 3/20 0.42
ALDH1A1 P00352 3/20 0.42
APOBEC3A P31941 1/20 0.42
APOBEC3G Q9HC16 1/20 0.42
SLC2A9 Q9NRM0 2/20 0.41
HTT P42858 1/20 0.41
IL15 P40933 1/20 0.41
IL2 P60568 1/20 0.41
IL15RA Q13261 1/20 0.41
KDM4E B2RXH2 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1719377 0.94 SLC22A12 (0.45) SLC22A12CYP2C9CYP2C19CYP1A2CYP3A4
SCHEMBL12010033 0.89 MAPT (0.47) SLC22A12CYP2C9CYP2C19CYP1A2CYP3A4
SCHEMBL250058 0.87 ALDH1A1 (0.43) SLC22A12CYP2C9CYP2C19CYP1A2CYP3A4
SCHEMBL29376753 0.84 SLC22A12 (0.65) SLC22A12CYP2C9CYP2C19CYP1A2CYP3A4
SCHEMBL248221 0.84 SLC22A12 (0.65) SLC22A12CYP2C9CYP2C19CYP1A2CYP3A4
SCHEMBL14921536 0.83 SLC22A12 (0.64) SLC22A12CYP2C9CYP2C19CYP1A2CYP3A4
Potassium SCHEMBL30892115 0.83 SLC22A12 (0.64) SLC22A12CYP2C9CYP2C19CYP1A2CYP3A4
SCHEMBL246489 0.81 CA1 (0.49) SLC22A12CYP2C9CYP2C19CYP1A2CYP3A4
SCHEMBL15556799 0.80 SLC22A12 (0.72) SLC22A12CYP2C9CYP2C19CYP1A2CYP3A4
SCHEMBL248911 0.79 MEN1 (0.48) KMT2AMEN1TDP1GAAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2402011-A1 Intermediates in the synthesis of S-triazolyl alpha-mercaptoacetanildes as inhibitors of HIV reverse transcriptase Ardea Biosciences, Inc. (US) 2012-01-04 EP disclosed