Croconazole

Croconazole

SCHEMBL34369

C=C(c1ccccc1OCc1cccc(Cl)c1)n1ccnc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR1I2 O75469 1/20 1.00
NR3C1 P04150 1/20 1.00
HTR1A P08908 1/20 1.00
ADORA3 P0DMS8 1/20 1.00
CNR1 P21554 1/20 1.00
TBXA2R P21731 1/20 1.00
SLC6A2 P23975 1/20 1.00
HTR2A P28223 1/20 1.00
HTR2C P28335 1/20 1.00
SLC6A4 P31645 1/20 1.00
ADRA1A P35348 1/20 1.00
OPRK1 P41145 1/20 1.00
HTR2B P41595 1/20 1.00
PDE4D Q08499 1/20 1.00
KCNH2 Q12809 1/20 1.00
ADRB2 P07550 10/20 0.53
ADRB1 P08588 10/20 0.53
ADRB3 P13945 10/20 0.53
SGMS2 Q8NHU3 1/20 0.51
ENPP2 Q13822 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Croconazole SCHEMBL7601955 1.00 NR1I2 (1.00) NR1I2NR3C1HTR1AADORA3CNR1
Croconazole SCHEMBL29378466 1.00 NR1I2 (1.00) NR1I2NR3C1HTR1AADORA3CNR1
Croconazole SCHEMBL36790 0.99 NR1I2 (0.98) NR1I2NR3C1HTR1AADORA3CNR1
Croconazole SCHEMBL121863 0.99 NR1I2 (0.98) NR1I2NR3C1HTR1AADORA3CNR1
Croconazole SCHEMBL1274172 0.93 NR1I2 (0.86) NR1I2NR3C1HTR1AADORA3CNR1
Croconazole SCHEMBL3690346 0.92 NR1I2 (0.85) NR1I2NR3C1HTR1AADORA3CNR1
SCHEMBL11090539 0.87 NR1I2 (0.78) NR1I2NR3C1HTR1AADORA3CNR1
SCHEMBL2449293 0.84 HTR1A (0.73) NR1I2NR3C1HTR1AADORA3CNR1
SCHEMBL2449294 0.84 HTR1A (0.73) NR1I2NR3C1HTR1AADORA3CNR1
SCHEMBL9662402 0.83 NR1I2 (0.72) NR1I2NR3C1HTR1AADORA3CNR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 4215 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12274830-B2 Nitric oxide inhalation therapy for infants with bronchiolitis BEYOND AIR LTD (IL) 2025-04-15 US claimed
US-20250099557-A1 ANTIBIOTIC PHARMACEUTICAL COMPOSITION CAPABLE OF SUBCUTANEOUS ADMINISTRATION SHANGHAI BAO PHARMACEUTICALS CO., LTD. (CN) 2025-03-27 US claimed
US-20250017904-A1 ANTIMICROBIAL COMPOSITIONS CONTAINING A SYNERGISTIC COMBINATION OF ACTIVATED CREATININE AND AN IMIDAZOLE ANTIFUNGAL AGENT BOARD OF REGENTS OF THE UNIVERSITY OF NEBRASKA (US) 2025-01-16 US claimed
WO-2024235510-A1 ANTI-DANDRUFF COMPOSITIONS ANALYTICON DISCOVERY GMBH (DE) 2024-11-21 WO claimed
EP-4464309-A1 ANTIDANDRUFF COMPOSITION COMPRISING 1-ACETOXYCHAVICOL ACETATE Analyticon Discovery GmbH (DE) 2024-11-20 EP claimed
US-20240173512-A1 METHODS FOR POTENTIATING ANTIMICROBIAL AGENTS STREETERVILLE CAPITAL, LLC 2024-05-30 US claimed
EP-4374848-A1 ANTIBIOTIC PHARMACEUTICAL COMPOSITION CAPABLE OF SUBCUTANEOUS ADMINISTRATION Shanghai Bao Pharmaceuticals Co., Ltd. (CN) 2024-05-29 EP claimed
WO-2024046311-A1 COMPOSITION USED FOR KILLING FUNGI AND METHOD FOR APPLYING COMPOSITION 江苏中旗科技股份有限公司 2024-03-07 WO claimed
US-11890421-B2 Methods for potentiating antimicrobial agents BEYOND AIR LTD (IL) 2024-02-06 US claimed
US-20230233483-A1 COMPOUND AND METHOD FOR THE TREATMENT OF CORONAVIRUSES APTEEUS (FR) 2023-07-27 US claimed
US-5374633-A Mixtures of nitrogen-heterocyclic antifungal compounds, fatty acid esters, propylene glycol and drugs, for increasing dosage by promoting absorption BRISTOL-MYERS SQUIBB COMPANY (US) 1994-12-20 US claimed
US-5214046-A Synergistic mixtures, inhibitors of sterol biosynthesis HOFFMANN-LA ROCHE INC. (US) 1993-05-25 US claimed
EP-0538442-A1 METHOD FOR IMPROVING THE THERAPEUTIC EFFICIENCY OF LIPOSOLUBLE ANTIFUNGAL AGENTS FROM THE IMIDAZOLE FAMILY, AND COMPOSITION FOR IMPLEMENTING SAME. OREAL (FR) 1993-04-28 EP claimed
WO-1992019225-A1 METHOD FOR IMPROVING THE THERAPEUTIC EFFICIENCY OF LIPOSOLUBLE ANTIFUNGAL AGENTS FROM THE IMIDAZOLE FAMILY, AND COMPOSITION FOR IMPLEMENTING SAME L'OREAL (FR) 1992-11-12 WO claimed
EP-0457333-A2 Topical composition Bristol-Myers Squibb Company (US) 1991-11-21 EP claimed
EP-0310122-B1 ANTIFUNGAL COMPOSITION KAKEN PHARMACEUTICAL CO., LTD. (JP) 1991-07-24 EP claimed
EP-0319965-B1 PHARMACEUTICAL PREPARATION FOR TINEA PEDIS SHIONOGI SEIYAKU KABUSHIKI KAISHA (JP) 1991-03-13 EP claimed
EP-0310122-A1 Antifungal composition KAKEN PHARMACEUTICAL CO., LTD. (JP) 1989-04-05 EP claimed
US-4483866-A FUNGICIDE SHIONOGI & CO., LTD. (JP) 1984-11-20 US claimed
US-4328348-A Novel benzylimidazole derivatives SHIONOGI & CO., LTD. (JP) 1982-05-04 US claimed