SCHEMBL3439643

SCHEMBL3439643

Cc1cc(N)c(Br)cc1N

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 4/20 0.63
TSHR P16473 3/20 0.63
MAPK1 P28482 1/20 0.63
ALDH1A1 P00352 7/20 0.50
CYP1A2 P05177 1/20 0.44
ALOX15 P16050 1/20 0.44
CASP7 P55210 1/20 0.44
HIF1A Q16665 1/20 0.44
HSD17B10 Q99714 1/20 0.44
POLB P06746 3/20 0.42
L3MBTL1 Q9Y468 2/20 0.42
TERT O14746 1/20 0.42
TDP1 Q9NUW8 4/20 0.42
CASP1 P29466 1/20 0.42
CD44 P16070 1/20 0.42
MAPT P10636 4/20 0.41
MEN1 O00255 1/20 0.41
APAF1 O14727 1/20 0.41
THRB P10828 1/20 0.41
NR4A1 P22736 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8121628 0.88 CYP3A4 (0.55) CYP3A4TSHRMAPK1ALDH1A1CYP1A2
SCHEMBL4508097 0.88 TSHR (0.63) CYP3A4TSHRMAPK1ALDH1A1CYP1A2
SCHEMBL9068413 0.86 CYP3A4 (0.46) CYP3A4TSHRMAPK1ALDH1A1CYP1A2
SCHEMBL2321600 0.86 CYP3A4 (0.52) CYP3A4TSHRMAPK1ALDH1A1CYP1A2
SCHEMBL17298241 0.85 CYP3A4 (0.58) CYP3A4TSHRMAPK1ALDH1A1CYP1A2
SCHEMBL33943 0.84 CYP3A4 (0.86) CYP3A4TSHRMAPK1ALDH1A1CYP1A2
SCHEMBL5519306 0.84 MAPT (0.50) CYP3A4TSHRMAPK1ALDH1A1ALOX15
SCHEMBL10620546 0.83 CYP3A4 (0.43) CYP3A4TSHRMAPK1ALDH1A1CYP1A2
Benzene SCHEMBL27906205 0.83 CYP3A4 (0.57) CYP3A4TSHRMAPK1ALDH1A1CYP1A2
SCHEMBL272760 0.82 CYP3A4 (0.63) CYP3A4TSHRMAPK1ALDH1A1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2402329-A1 Analgetic phenylsulphonamides Boehringer Ingelheim International GmbH (DE) 2012-01-04 EP disclosed