SCHEMBL3440809

SCHEMBL3440809

C[C@@]12CCC[C@H]1[C@@H]1CCC3C[C@@H](O)CC[C@]3(C)[C@H]1CC2

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR1I3 Q14994 1/20 1.00
CDK5 Q00535 1/20 0.70
CDK5R1 Q15078 1/20 0.70
LMNA P02545 3/20 0.67
GPBAR1 Q8TDU6 2/20 0.67
CYP3A4 P08684 2/20 0.67
SHBG P04278 1/20 0.67
SERPINA6 P08185 1/20 0.67
CYP1A2 P05177 1/20 0.67
CYP2C9 P11712 1/20 0.67
TSHR P16473 1/20 0.67
CYP2C19 P33261 1/20 0.67
HSD17B10 Q99714 1/20 0.67
GRIN1 Q05586 2/20 0.63
GRIN2B Q13224 2/20 0.63
G6PD P11413 2/20 0.59
MEN1 O00255 1/20 0.59
GABRP O00591 1/20 0.59
GABRD O14764 1/20 0.59
GMNN O75496 1/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1047682 1.00 NR1I3 (1.00) NR1I3CDK5CDK5R1LMNAGPBAR1
SCHEMBL15963473 1.00 NR1I3 (1.00) NR1I3CDK5CDK5R1LMNAGPBAR1
SCHEMBL3130550 1.00 NR1I3 (1.00) NR1I3CDK5CDK5R1LMNAGPBAR1
SCHEMBL2555591 1.00 NR1I3 (1.00) NR1I3CDK5CDK5R1LMNAGPBAR1
SCHEMBL13785427 1.00 NR1I3 (1.00) NR1I3CDK5CDK5R1LMNAGPBAR1
SCHEMBL11128263 1.00 NR1I3 (1.00) NR1I3CDK5CDK5R1LMNAGPBAR1
SCHEMBL21802632 1.00 NR1I3 (1.00) NR1I3CDK5CDK5R1LMNAGPBAR1
SCHEMBL20781172 1.00 NR1I3 (1.00) NR1I3CDK5CDK5R1LMNAGPBAR1
SCHEMBL20781187 1.00 NR1I3 (1.00) NR1I3CDK5CDK5R1LMNAGPBAR1
SCHEMBL11250886 1.00 NR1I3 (1.00) NR1I3CDK5CDK5R1LMNAGPBAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108084239-A The preparation method of (3 β, 15 α)--14 β of dihydroxy-phenylamino or benzyl amino androstane -17- ketone 扬州大学 2018-05-29 CN claimed
CN-105693801-B The aryl androstane 5 (6), 8 (14) of 3 β hydroxyls 16, the synthetic method of the ketone of 15 (16) triolefin 17 泰州职业技术学院 2017-05-31 CN claimed
EP-2206719-A2 Novel C-17-Heteroaryl Steroidal CYP17 Inhibitors/Antiandrogens: Synthesis, In Vitro Biological Activities, Pharmacokinetics and Antitumor University Of Maryland (US) 2010-07-14 EP claimed
CN-108084239-A The preparation method of (3 β, 15 α)--14 β of dihydroxy-phenylamino or benzyl amino androstane -17- ketone 扬州大学 2018-05-29 CN disclosed
EP-3186267-A1 AMPHIPHILIC COMPOUNDS WITH NEUROPROTECTIVE PROPERTIES Ustav Organicke Chemie a Biochemie AV CR, v.v.i. (CZ) 2017-07-05 EP disclosed
CN-105732755-B The aryl androstane 5 (6), 8 (14) of 3 β hydroxyls 16, the ketone of 15 (16) triolefin 17 泰州职业技术学院 2017-05-31 CN disclosed
CN-105693801-B The aryl androstane 5 (6), 8 (14) of 3 β hydroxyls 16, the synthetic method of the ketone of 15 (16) triolefin 17 泰州职业技术学院 2017-05-31 CN disclosed
WO-2016029888-A1 AMPHIPHILIC COMPOUNDS WITH NEUROPROTECTIVE PROPERTIES USTAV ORGANICKE CHEMIE A BIOCHEMIE AV CR, V.V.I. (CZ) 2016-03-03 WO disclosed
WO-2015003003-A1 SHIP INHIBITION TO COMBAT OBESITY THE RESEARCH FOUNDATION FOR THE STATE UNIVERSITY OF NEW YORK (US) 2015-01-08 WO disclosed
CN-1501795-A Gaba-receptor modulators for the treatment of neurodegenerative diseases of the eye ��������²�ʿ��ѧҩ������ɷ����� 2004-06-02 CN disclosed