SCHEMBL3441226

SCHEMBL3441226

COC(=O)Oc1cc(N)ccn1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.39
KDM4C Q9H3R0 2/20 0.38
AAK1 Q2M2I8 1/20 0.38
ALDH1A1 P00352 3/20 0.36
LOX P28300 1/20 0.36
LOXL2 Q9Y4K0 1/20 0.36
ACACB O00763 2/20 0.36
KDM4E B2RXH2 3/20 0.36
KDM6B O15054 1/20 0.36
KDM5C P41229 1/20 0.36
KDM2A Q9Y2K7 1/20 0.36
KDM3A Q9Y4C1 1/20 0.36
ALOX5 P09917 1/20 0.36
NOS3 P29474 1/20 0.35
NOS1 P29475 1/20 0.35
NOS2 P35228 1/20 0.35
HPGD P15428 1/20 0.35
HSD17B10 Q99714 1/20 0.35
GABRP O00591 1/20 0.34
GABRD O14764 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9568958 0.82 AAK1 (0.38) KDM4CAAK1ALDH1A1ACACBKDM4E
SCHEMBL27837097 0.81 CYP19A1 (0.40) GAAKDM4CALDH1A1LOXLOXL2
SCHEMBL25984978 0.81 KDM4C (0.44) KDM4CAAK1ALDH1A1ACACBNOS1
SCHEMBL2920954 0.81 KDM4E (0.44) GAAKDM4CAAK1ALDH1A1ACACB
SCHEMBL22946357 0.78 MEN1 (0.40) GAAKDM4CALDH1A1ACACBKDM4E
SCHEMBL9573013 0.78 KDM4E (0.36) KDM4CAAK1ALDH1A1ACACBKDM4E
SCHEMBL22557503 0.77 ESR1 (0.39) KDM4CLOXLOXL2NOS3NOS1
SCHEMBL7871639 0.77 AAK1 (0.35) KDM4CAAK1ALDH1A1ACACBKDM4E
SCHEMBL22952872 0.76 SMN1; SMN2 (0.43) ALDH1A1KDM4E
SCHEMBL9018039 0.75 KDM4E (0.44) ALDH1A1ACACBKDM4EHPGDHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010133312-A1 HALOGEN-SUBSTITUTED COMPOUNDS AS PESTICIDES BAYER CROPSCIENCE AKTIENGESELLSCHAFT (DE) 2010-11-25 WO disclosed
EP-2253617-A1 Halogenated compounds as pesticides Bayer CropScience AG (DE) 2010-11-24 EP disclosed
EP-1202988-A2 NOVEL INTEGRIN RECEPTOR ANTAGONISTS BASF AKTIENGESELLSCHAFT (DE) 2002-05-08 EP disclosed
EP-1173468-A1 INTEGRIN RECEPTOR ANTAGONISTS BASF AKTIENGESELLSCHAFT (DE) 2002-01-23 EP disclosed
WO-2001010847-A2 NOVEL INTEGRIN RECEPTOR ANTAGONISTS BASF AKTIENGESELLSCHAFT (DE) 2001-02-15 WO disclosed
WO-2000066618-A1 INTEGRIN RECEPTOR ANTAGONISTS BASF AKTIENGESELLSCHAFT (DE) 2000-11-09 WO disclosed