SCHEMBL9568958

SCHEMBL9568958

COC(=O)Oc1ccnc(OC(=O)OC)c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AAK1 Q2M2I8 1/20 0.38
CCR1 P32246 1/20 0.37
CCR5 P51681 1/20 0.37
CCR8 P51685 1/20 0.37
RIOK2 Q9BVS4 1/20 0.36
ACACB O00763 6/20 0.36
KDM4E B2RXH2 2/20 0.36
KDM6B O15054 1/20 0.36
KDM5C P41229 1/20 0.36
KDM4C Q9H3R0 1/20 0.36
KDM2A Q9Y2K7 1/20 0.36
KDM3A Q9Y4C1 1/20 0.36
NOS3 P29474 1/20 0.35
NOS1 P29475 1/20 0.35
NOS2 P35228 1/20 0.35
HPGD P15428 1/20 0.35
HSD17B10 Q99714 1/20 0.35
KMT2A Q03164 2/20 0.35
ALDH1A1 P00352 1/20 0.35
MEN1 O00255 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9573013 0.92 KDM4E (0.36) AAK1CCR1CCR5CCR8RIOK2
SCHEMBL7871639 0.90 AAK1 (0.35) AAK1CCR1CCR5CCR8RIOK2
SCHEMBL19664383 0.85 ACACB (0.36) ACACBKMT2AALDH1A1MEN1
SCHEMBL9706059 0.84 MEN1 (0.49) ACACBHPGDHSD17B10KMT2AALDH1A1
SCHEMBL2549948 0.84 CCR1 (0.57) CCR1CCR5CCR8RIOK2KDM4E
SCHEMBL9662430 0.83 LMNA (0.36) AAK1HSD17B10KMT2AALDH1A1
SCHEMBL3441226 0.82 GAA (0.39) AAK1ACACBKDM4EKDM6BKDM5C
SCHEMBL9706023 0.82 LOXL2 (0.46) HPGD
SCHEMBL19664384 0.81 KMT2A (0.45) KDM4ENOS3NOS1NOS2KMT2A
SCHEMBL9663046 0.81 TSHR (0.38) AAK1ACACBKDM4ENOS2KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2861206-B1 COMPOSITION INCLUDING A PYRIDINE DICARBOXYLIC ACID ESTER AND A BINDING POLYMER, METHOD THEREFOR, AND USE THEREOF FOR TREATING HAIR OREAL (FR) 2019-06-12 EP claimed
EP-2861205-B1 COMPOSITION INCLUDING A PYRIDINE DICARBOXYLIC ACID ESTER AND A GLUCOSE AND FATTY ACID ESTER. OREAL (FR) 2017-12-06 EP claimed
EP-0548883-A1 Substituted pyridine-N-oxides, process for their preparation and their use as medicines HOECHST AKTIENGESELLSCHAFT (DE) 1993-06-30 EP disclosed
EP-0541042-A1 2,4- and 2,5-pyridine-dicarboxylic acid derivatives, process for their preparation and their use HOECHST AKTIENGESELLSCHAFT (DE) 1993-05-12 EP disclosed