SCHEMBL3445000

SCHEMBL3445000

CC(O)CNc1nc(NCc2ccc(Cl)c(N)c2)c2nnn(C(C)C)c2n1

nearest known ligand 0.47

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CDK2 P24941 8/20 0.47
CDK1 P06493 3/20 0.47
CDK9 P50750 2/20 0.44
BCDIN3D Q7Z5W3 8/20 0.41
CCNE1 P24864 5/20 0.41
CDK5 Q00535 1/20 0.39
CCNE2 O96020 3/20 0.39
CCNA2 P20248 1/20 0.39
CCNA1 P78396 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3445582 0.92 BCDIN3D (0.50) CDK2CDK1BCDIN3DCCNE1CDK5
SCHEMBL3445297 0.90 BCDIN3D (0.46) CDK2CDK1CDK9BCDIN3DCCNE1
SCHEMBL3446859 0.88 CDK2 (0.44) CDK2CDK1CDK9BCDIN3DCCNE1
SCHEMBL3444468 0.86 FLT3 (0.47) CDK2CDK1CDK9BCDIN3DCCNE1
SCHEMBL3444370 0.85 CDK2 (0.54) CDK2CDK1CDK9CCNE1CDK5
SCHEMBL3444366 0.85 CDK2 (0.54) CDK2CDK1CDK9CCNE1CDK5
SCHEMBL3445110 0.84 CDK2 (0.55) CDK2CDK1CDK9CCNE1CDK5
SCHEMBL6203983 0.84 KMT2A (0.42) CDK1BCDIN3DCDK5
SCHEMBL3444838 0.83 CDK2 (0.45) CDK2CDK1CDK9CCNE1CDK5
SCHEMBL3446716 0.82 CDK2 (0.67) CDK2CDK1CDK9CCNE1CDK5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7816350-B2 Substituted [1,2,3] triazolo[4,5-D]pyrimidines as cdk inhibitors INSTITUTE OF EXPERIMENTAL BOTANY ASCR (CZ) 2010-10-19 US claimed