SCHEMBL6203983

SCHEMBL6203983

CC(C)c1nc(NCc2ccc(Cl)c(N)c2)c2nnn(C(C)C)c2n1

nearest known ligand 0.42

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 1/20 0.42
ALDH1A1 P00352 1/20 0.38
LMNA P02545 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
CDK1 P06493 3/20 0.37
CCNB2 O95067 1/20 0.37
CCNB1 P14635 1/20 0.37
CDK5 Q00535 1/20 0.37
CCNB3 Q8WWL7 1/20 0.37
GAA P10253 1/20 0.36
TRPV1 Q8NER1 1/20 0.36
CTSL P07711 6/20 0.35
RAB9A P51151 1/20 0.35
PDE8B O95263 1/20 0.34
BCDIN3D Q7Z5W3 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3445582 0.84 BCDIN3D (0.50) CDK1CDK5BCDIN3D
SCHEMBL3445000 0.84 CDK2 (0.47) CDK1CDK5BCDIN3D
SCHEMBL3444366 0.81 CDK2 (0.54) KMT2AALDH1A1CDK1CCNB2CCNB1
SCHEMBL3444370 0.81 CDK2 (0.54) KMT2AALDH1A1CDK1CCNB2CCNB1
SCHEMBL3445110 0.81 CDK2 (0.55) ALDH1A1LMNASMN1; SMN2CDK1CCNB2
SCHEMBL6226169 0.80 KMT2A (0.56) KMT2AALDH1A1LMNASMN1; SMN2CDK1
SCHEMBL3445180 0.80 CCNE1 (0.55) CDK5
SCHEMBL6201910 0.79 ALDH1A1 (0.49) KMT2AALDH1A1LMNASMN1; SMN2CDK1
SCHEMBL3445887 0.79 CDK2 (0.53) CDK1CCNB1CDK5RAB9ABCDIN3D
SCHEMBL6203832 0.76 KMT2A (0.46) KMT2AALDH1A1LMNASMN1; SMN2CDK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1539760-A2 AZAPURINE DERIVATIVES INSTITUTE OF EXPERIMENTAL BOTANY ASCR (CZ) 2005-06-15 EP claimed
WO-2004018473-A2 AZAPURINE DERIVATIVES INSTITUTE OF EXPERIMENTAL BOTANY ASCR (CZ) 2004-03-04 WO claimed
EP-1539760-A2 AZAPURINE DERIVATIVES INSTITUTE OF EXPERIMENTAL BOTANY ASCR (CZ) 2005-06-15 EP disclosed
WO-2004018473-A2 AZAPURINE DERIVATIVES INSTITUTE OF EXPERIMENTAL BOTANY ASCR (CZ) 2004-03-04 WO disclosed