SCHEMBL3445168

SCHEMBL3445168

CCC(CO)Nc1nc(NCc2c(O)cc(OC)cc2O)c2nnn(C(C)C)c2n1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK1 P06493 12/20 0.49
CCNB1 P14635 5/20 0.49
CCNB2 O95067 4/20 0.49
CCNB3 Q8WWL7 4/20 0.49
CDK2 P24941 11/20 0.47
CCNE1 P24864 10/20 0.47
CDK9 P50750 7/20 0.47
CCNT1 O60563 5/20 0.47
CCNE2 O96020 2/20 0.47
CCNT2 O60583 1/20 0.47
CDK5 Q00535 6/20 0.47
CDK5R1 Q15078 4/20 0.47
CACNA1B Q00975 2/20 0.47
CCNK O75909 2/20 0.46
CDK12 Q9NYV4 2/20 0.46
CDK7 P50613 4/20 0.45
CSNK1D P48730 2/20 0.45
CLK2 P49760 2/20 0.45
CSNK1G2 P78368 2/20 0.45
DYRK1A Q13627 2/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3446297 0.89 CDK1 (0.46) CDK1CCNB1CCNB2CCNB3CDK2
SCHEMBL3445759 0.89 CDK2 (0.54) CDK1CCNB1CCNB2CCNB3CDK2
SCHEMBL3446158 0.88 CDK1 (0.48) CDK1CCNB1CCNB2CCNB3CDK2
SCHEMBL3446165 0.88 CDK1 (0.48) CDK1CCNB1CCNB2CCNB3CDK2
SCHEMBL3445194 0.88 CDK1 (0.45) CDK1CCNB1CCNB2CCNB3CDK2
SCHEMBL3444719 0.84 CDK2 (0.55) CDK1CCNB1CCNB2CCNB3CDK2
SCHEMBL3445883 0.83 CDK2 (0.42) CDK1CDK2CCNE1CDK9CCNT1
SCHEMBL3446276 0.83 CDK2 (0.40) CDK1CDK2CCNE1CDK9CCNT1
SCHEMBL3445192 0.81 CDK1 (0.72) CDK1CCNB1CCNB2CCNB3CDK2
SCHEMBL3446739 0.81 CDK2 (0.62) CDK1CCNB1CCNB2CCNB3CDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7816350-B2 Substituted [1,2,3] triazolo[4,5-D]pyrimidines as cdk inhibitors INSTITUTE OF EXPERIMENTAL BOTANY ASCR (CZ) 2010-10-19 US claimed