SCHEMBL3445585

SCHEMBL3445585

CCn1nnc2c(NCc3cccc(OC(C)=O)c3)nc(NCC(C)O)nc21

nearest known ligand 0.46

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CDK2 P24941 8/20 0.46
CDK1 P06493 6/20 0.46
CDK9 P50750 4/20 0.43
CCNE1 P24864 4/20 0.39
CDK5 Q00535 2/20 0.39
CCNE2 O96020 1/20 0.37
CCNB2 O95067 1/20 0.37
CCNB1 P14635 1/20 0.37
CCNB3 Q8WWL7 1/20 0.37
CDK7 P50613 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
KDM4E B2RXH2 1/20 0.36
NPC1 O15118 1/20 0.36
MAPT P10636 1/20 0.36
TDP1 Q9NUW8 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3446713 0.92 CDK2 (0.41) CDK2CDK1CDK9CCNE1CDK5
SCHEMBL3445601 0.90 CDK2 (0.47) CDK2CDK1CDK9CCNE1CDK5
SCHEMBL3445310 0.89 CDK2 (0.49) CDK2CDK1CDK9CCNE1CDK5
SCHEMBL3446243 0.86 CDK1 (0.51) CDK2CDK1CDK9CCNE1CDK5
SCHEMBL3446242 0.86 CDK1 (0.51) CDK2CDK1CDK9CCNE1CDK5
SCHEMBL3445495 0.85 CDK1 (0.51) CDK2CDK1CDK9CCNE1CDK5
SCHEMBL3445451 0.84 CDK2 (0.43) CDK2CDK1CDK9CCNE1CDK5
SCHEMBL3455226 0.84 CDK2 (0.63) CDK2CDK1CDK9CCNE1CDK5
SCHEMBL3445798 0.82 BCDIN3D (0.43) CDK2CDK1CDK9CCNE1CDK5
SCHEMBL3445863 0.81 CDK2 (0.49) CDK2CDK1CDK9CCNE1CDK5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7816350-B2 Substituted [1,2,3] triazolo[4,5-D]pyrimidines as cdk inhibitors INSTITUTE OF EXPERIMENTAL BOTANY ASCR (CZ) 2010-10-19 US claimed