SCHEMBL3445451

SCHEMBL3445451

CCn1nnc2c(NCc3ccccc3OC(C)=O)nc(NCC(C)O)nc21

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK2 P24941 6/20 0.43
CCNE1 P24864 3/20 0.43
CDK1 P06493 6/20 0.43
CDK9 P50750 3/20 0.40
CDK5 Q00535 3/20 0.40
CCNT1 O60563 1/20 0.40
CDK5R1 Q15078 1/20 0.40
ALDH1A1 P00352 2/20 0.39
MAPT P10636 1/20 0.39
PKM P14618 1/20 0.39
TSHR P16473 1/20 0.39
HTT P42858 1/20 0.39
POLB P06746 1/20 0.38
LMNA P02545 1/20 0.37
JAK1 P23458 1/20 0.36
JAK3 P52333 1/20 0.36
CDK7 P50613 1/20 0.35
GBA1 P04062 1/20 0.35
CCNB2 O95067 1/20 0.35
CCNB1 P14635 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3445266 0.92 CDK2 (0.40) CDK2CCNE1CDK1CDK9CDK5
SCHEMBL3445433 0.89 POLB (0.47) CDK2CCNE1CDK1CDK9CDK5
SCHEMBL3446366 0.89 CDK2 (0.46) CDK2CCNE1CDK1CDK9CDK5
SCHEMBL3445734 0.85 CDK1 (0.49) CDK2CCNE1CDK1CDK9CDK5
SCHEMBL3445739 0.85 CDK1 (0.49) CDK2CCNE1CDK1CDK9CDK5
SCHEMBL3446533 0.84 CDK2 (0.49) CDK2CCNE1CDK1CDK9CDK5
SCHEMBL3445585 0.84 CDK2 (0.46) CDK2CCNE1CDK1CDK9CDK5
SCHEMBL3445380 0.83 CDK2 (0.61) CDK2CCNE1CDK1CDK9CDK5
SCHEMBL3446329 0.83 CDK2 (0.51) CDK2CCNE1CDK1CDK9CDK5
SCHEMBL3446876 0.81 POLB (0.46) CDK2CCNE1CDK1CDK9CDK5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7816350-B2 Substituted [1,2,3] triazolo[4,5-D]pyrimidines as cdk inhibitors INSTITUTE OF EXPERIMENTAL BOTANY ASCR (CZ) 2010-10-19 US claimed