SCHEMBL3445693

SCHEMBL3445693

CC(O)CNc1nc(NCc2cc(O)c(Cl)cc2O)c2nnn(C)c2n1

nearest known ligand 0.41

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CDK2 P24941 12/20 0.41
CCNE1 P24864 10/20 0.41
CDK5 Q00535 7/20 0.41
CDK5R1 Q15078 7/20 0.41
CDK7 P50613 5/20 0.41
CCNH P51946 5/20 0.41
CDK1 P06493 2/20 0.41
CDK9 P50750 8/20 0.40
CCNT1 O60563 7/20 0.40
CCNT2 O60583 1/20 0.40
CCNE2 O96020 1/20 0.40
BCDIN3D Q7Z5W3 3/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3445470 0.91 BCDIN3D (0.44) CDK2CCNE1CDK5CDK5R1CDK7
SCHEMBL3446239 0.89 CDK2 (0.43) CDK2CCNE1CDK5CDK5R1CDK7
SCHEMBL3444559 0.89 CDK2 (0.41) CDK2CCNE1CDK5CDK5R1CDK7
SCHEMBL3446232 0.87 POLB (0.44) CDK2CCNE1CDK5CDK5R1CDK7
SCHEMBL3445466 0.85 CDK1 (0.50) CDK2CCNE1CDK5CDK5R1CDK7
SCHEMBL3445465 0.85 CDK1 (0.50) CDK2CCNE1CDK5CDK5R1CDK7
SCHEMBL3455221 0.84 CDK2 (0.43) CDK2CCNE1CDK5CDK5R1CDK7
SCHEMBL3444444 0.84 CDK2 (0.42) CDK2CCNE1CDK5CDK5R1CDK7
SCHEMBL3445471 0.82 CDK2 (0.56) CDK2CCNE1CDK5CDK5R1CDK7
SCHEMBL3445769 0.81 CDK2 (0.42) CDK2CCNE1CDK5CDK5R1CDK7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7816350-B2 Substituted [1,2,3] triazolo[4,5-D]pyrimidines as cdk inhibitors INSTITUTE OF EXPERIMENTAL BOTANY ASCR (CZ) 2010-10-19 US claimed