SCHEMBL3446239

SCHEMBL3446239

CC(O)CNc1nc(NCc2cc(O)c(Cl)cc2O)c2nnn(C(C)C)c2n1

nearest known ligand 0.43

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CDK2 P24941 14/20 0.43
CCNE1 P24864 11/20 0.43
CDK5 Q00535 8/20 0.43
CDK5R1 Q15078 8/20 0.43
CDK7 P50613 5/20 0.43
CCNH P51946 5/20 0.43
CDK1 P06493 3/20 0.42
CDK9 P50750 9/20 0.42
CCNT1 O60563 8/20 0.42
CCNT2 O60583 1/20 0.42
CCNE2 O96020 1/20 0.42
FLT3 P36888 1/20 0.36
CCNB2 O95067 1/20 0.35
CCNB1 P14635 1/20 0.35
CCNB3 Q8WWL7 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3445769 0.91 CDK2 (0.42) CDK2CCNE1CDK5CDK5R1CDK7
SCHEMBL3445693 0.89 CDK2 (0.41) CDK2CCNE1CDK5CDK5R1CDK7
SCHEMBL3444559 0.88 CDK2 (0.41) CDK2CCNE1CDK5CDK5R1CDK7
SCHEMBL3445754 0.87 CDK2 (0.41) CDK2CCNE1CDK5CDK5R1CDK7
SCHEMBL3446759 0.85 CDK2 (0.44) CDK2CCNE1CDK5CDK5R1CDK7
SCHEMBL3446389 0.84 CDK2 (0.43) CDK2CCNE1CDK5CDK5R1CDK7
SCHEMBL3446471 0.84 CDK1 (0.51) CDK2CCNE1CDK5CDK5R1CDK7
SCHEMBL3446473 0.84 CDK1 (0.51) CDK2CCNE1CDK5CDK5R1CDK7
SCHEMBL3444987 0.83 CDK2 (0.59) CDK2CCNE1CDK5CDK5R1CDK7
SCHEMBL3445143 0.81 CCNE1 (0.61) CDK2CCNE1CDK5CDK5R1CDK7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7816350-B2 Substituted [1,2,3] triazolo[4,5-D]pyrimidines as cdk inhibitors INSTITUTE OF EXPERIMENTAL BOTANY ASCR (CZ) 2010-10-19 US claimed