SCHEMBL3445732

SCHEMBL3445732

CC(O)CNc1nc(Nc2ccc(Br)cc2)c2nnn(C)c2n1

nearest known ligand 0.66

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
FLT3 P36888 7/20 0.66
CDK2 P24941 3/20 0.47
CCNE2 O96020 2/20 0.47
CCNE1 P24864 2/20 0.47
CDK1 P06493 4/20 0.46
KDM4E B2RXH2 1/20 0.44
MEN1 O00255 1/20 0.44
ALDH1A1 P00352 1/20 0.44
MAPT P10636 1/20 0.44
MAPK1 P28482 1/20 0.44
KMT2A Q03164 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44
BCDIN3D Q7Z5W3 4/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3446225 0.89 FLT3 (0.60) FLT3CDK2CCNE1CDK1KDM4E
SCHEMBL3446050 0.89 FLT3 (0.53) FLT3CDK2CCNE2CCNE1CDK1
SCHEMBL3445068 0.89 FLT3 (0.54) FLT3CDK2CDK1MAPTBCDIN3D
SCHEMBL3446201 0.88 FLT3 (0.68) FLT3CDK2CCNE2CCNE1CDK1
SCHEMBL3444510 0.87 FLT3 (0.64) FLT3CDK2CCNE2CCNE1CDK1
SCHEMBL3445097 0.82 FLT3 (0.46) FLT3CDK1MEN1KMT2ABCDIN3D
SCHEMBL3445721 0.82 FLT3 (0.46) FLT3CDK2CCNE2CCNE1CDK1
SCHEMBL3445655 0.82 CDK1 (0.68) CDK2CCNE2CCNE1CDK1KDM4E
SCHEMBL3445657 0.82 CDK1 (0.68) CDK2CCNE2CCNE1CDK1KDM4E
SCHEMBL3445090 0.81 CDK1 (0.53) FLT3CDK2CCNE2CCNE1CDK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7816350-B2 Substituted [1,2,3] triazolo[4,5-D]pyrimidines as cdk inhibitors INSTITUTE OF EXPERIMENTAL BOTANY ASCR (CZ) 2010-10-19 US claimed