SCHEMBL3445752

SCHEMBL3445752

CCC(CO)Nc1nc(Nc2cccc(Cl)c2)c2nnn(C(C)C)c2n1

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK5 Q00535 14/20 0.71
CDK5R1 Q15078 13/20 0.71
KDM4E B2RXH2 4/20 0.71
MAPT P10636 3/20 0.71
NPC1 O15118 1/20 0.71
POLB P06746 1/20 0.71
NPSR1 Q6W5P4 1/20 0.60
TDP1 Q9NUW8 1/20 0.60
CDK1 P06493 6/20 0.56
CCNA2 P20248 11/20 0.55
CDK2 P24941 11/20 0.55
CCNA1 P78396 10/20 0.55
DYRK1A Q13627 10/20 0.55
CCNB1 P14635 3/20 0.55
CCNE1 P24864 2/20 0.55
MAPK1 P28482 2/20 0.55
MEN1 O00255 1/20 0.55
CCNB2 O95067 1/20 0.55
PAK4 O96013 1/20 0.55
CCNE2 O96020 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3446331 0.89 CDK5 (0.68) CDK5CDK5R1KDM4EMAPTNPC1
SCHEMBL3444971 0.89 CDK5 (0.55) CDK5CDK5R1KDM4EMAPTNPC1
SCHEMBL3446637 0.88 CDK5 (0.56) CDK5CDK5R1KDM4EMAPTNPC1
SCHEMBL3445128 0.88 CDK1 (0.72) CDK5CDK5R1KDM4EMAPTNPC1
SCHEMBL3445426 0.88 CDK5 (0.67) CDK5CDK5R1KDM4EMAPTNPC1
SCHEMBL3445316 0.88 CDK1 (0.72) CDK5CDK5R1KDM4EMAPTNPC1
SCHEMBL3445575 0.87 CDK1 (0.55) CDK5CDK5R1KDM4EMAPTNPC1
SCHEMBL3445857 0.85 CDK5 (0.53) CDK5CDK5R1KDM4EMAPTNPC1
SCHEMBL3446513 0.85 CDK5 (0.53) CDK5CDK5R1KDM4EMAPTNPC1
SCHEMBL3444661 0.83 CDK5 (0.58) CDK5CDK5R1KDM4EMAPTNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7816350-B2 Substituted [1,2,3] triazolo[4,5-D]pyrimidines as cdk inhibitors INSTITUTE OF EXPERIMENTAL BOTANY ASCR (CZ) 2010-10-19 US claimed