SCHEMBL3445857

SCHEMBL3445857

CCC(CO)Nc1nc(Nc2ccc(N)c(Cl)c2)c2nnn(C(C)C)c2n1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK5 Q00535 16/20 0.53
CDK5R1 Q15078 15/20 0.53
KDM4E B2RXH2 2/20 0.53
MAPT P10636 2/20 0.53
NPC1 O15118 1/20 0.53
POLB P06746 1/20 0.53
CDK2 P24941 15/20 0.48
CCNA2 P20248 14/20 0.48
CCNA1 P78396 13/20 0.48
DYRK1A Q13627 13/20 0.48
CDK1 P06493 4/20 0.45
CSNK1A1 P48729 2/20 0.45
CCNE1 P24864 2/20 0.45
CCNT1 O60563 1/20 0.45
CCNB1 P14635 1/20 0.45
CDK7 P50613 1/20 0.45
CDK9 P50750 1/20 0.45
CCNH P51946 1/20 0.45
MNAT1 P51948 1/20 0.45
GSK3B P49841 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3446513 0.93 CDK5 (0.53) CDK5CDK5R1KDM4EMAPTNPC1
SCHEMBL3445806 0.89 CDK5 (0.50) CDK5CDK5R1KDM4EMAPTNPC1
SCHEMBL3446747 0.88 CDK5 (0.49) CDK5CDK5R1KDM4EMAPTNPC1
SCHEMBL3444524 0.88 CDK5 (0.55) CDK5CDK5R1KDM4EMAPTCDK2
SCHEMBL3444523 0.88 CDK5 (0.55) CDK5CDK5R1KDM4EMAPTCDK2
SCHEMBL3444661 0.87 CDK5 (0.58) CDK5CDK5R1KDM4EMAPTNPC1
SCHEMBL3444971 0.87 CDK5 (0.55) CDK5CDK5R1KDM4EMAPTNPC1
SCHEMBL3445575 0.85 CDK1 (0.55) CDK5CDK5R1KDM4EMAPTNPC1
SCHEMBL3445752 0.85 CDK5 (0.71) CDK5CDK5R1KDM4EMAPTNPC1
SCHEMBL3446427 0.83 CDK5 (0.55) CDK5CDK5R1KDM4EMAPTNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7816350-B2 Substituted [1,2,3] triazolo[4,5-D]pyrimidines as cdk inhibitors INSTITUTE OF EXPERIMENTAL BOTANY ASCR (CZ) 2010-10-19 US claimed